SCHEMBL9869213

SCHEMBL9869213

CCOC(=O)c1ccc(COC)nc1C(=O)OCC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.46
CA2 P00918 4/20 0.46
CA7 P43166 4/20 0.46
CA9 Q16790 4/20 0.46
CA14 Q9ULX7 4/20 0.46
CA1 P00915 3/20 0.46
TSHR P16473 2/20 0.46
KDM4E B2RXH2 3/20 0.43
HSD17B10 Q99714 2/20 0.43
CYP1A2 P05177 1/20 0.42
ALDH1A1 P00352 3/20 0.41
MAOB P27338 2/20 0.41
HPGD P15428 2/20 0.41
MIF P14174 1/20 0.41
PFKFB3 Q16875 1/20 0.41
MAOA P21397 1/20 0.41
TARBP2 Q15633 2/20 0.40
GABRP O00591 1/20 0.40
GABRD O14764 1/20 0.40
GABRA1 P14867 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9869056 0.88 CA12 (0.46) CA12CA2CA7CA9CA14
SCHEMBL9308690 0.86 TSHR (0.50) CA12CA2CA7CA9CA14
SCHEMBL9869721 0.82 TSHR (0.50) TSHRCYP1A2ALDH1A1MAOBGAA
SCHEMBL9308330 0.79 TSHR (0.53) CA12CA2CA7CA9CA14
SCHEMBL6306356 0.76 TSHR (0.50) CA12CA2CA7CA9CA14
SCHEMBL9869186 0.75 CA12 (0.42) CA12CA2CA7CA9CA14
SCHEMBL9869495 0.75 CA12 (0.42) CA12CA2CA7CA9CA14
SCHEMBL9315811 0.75 ALOX15 (0.45) CA12CA2CA7CA9CA14
SCHEMBL9869319 0.74 POLB (0.41) TSHRKDM4ECYP1A2ALDH1A1HPGD
SCHEMBL21371248 0.74 CYP1A2 (0.70) CA12CA2CA7CA9CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5041552-A Treatment of hypertension, heart failure, glaucoma and hyperaldosteronism WARNER-LAMBERT COMPANY (US) 1991-08-20 US disclosed
US-4997947-A Forming 6-substituted pyridine-2,3-dicarboxylic esters followed by reacting with aminoalkanecarboxylic acid amide; herbicides, plant growth regulators CIBA-GEIGY CORPORATION (US) 1991-03-05 US disclosed