SCHEMBL9869750

SCHEMBL9869750

CNS(=O)(=O)c1cc(C(=O)NC(CC2CC2)C2CCCN2)c2c(c1N)CCCO2

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 2/20 0.30
HTR1A P08908 1/20 0.30
ADRA2C P18825 1/20 0.30
ACHE P22303 1/20 0.30
PTGS1 P23219 1/20 0.30
ADRA1A P35348 1/20 0.30
HTR3A P46098 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9866623 0.99
SCHEMBL9866772 0.91 HTR4 (0.30) HTR4HTR1AADRA2CACHEPTGS1
SCHEMBL9868594 0.84 BACE1 (0.30)
SCHEMBL10561655 0.77 DRD2 (0.42) HTR4ADRA2CACHEHTR3AKCNH2
SCHEMBL9822959 0.77 DRD2 (0.30)
Hydrochloric Acid SCHEMBL9868759 0.77 BACE1 (0.31)
SCHEMBL9868848 0.76 BACE1 (0.33)
SCHEMBL9823201 0.76
SCHEMBL9867269 0.73 APP (0.34) HTR4HTR3A
SCHEMBL9869736 0.73 DRD2 (0.45) ADRA2CKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5006570-A Dihydrobenzofuran- and chroman-carboxamide derivatives, processes for the preparation thereof and use thereof as neuroleptics LABORATOIRES DELAGRANGE (FR) 1991-04-09 US disclosed