SCHEMBL9866772

SCHEMBL9866772

CCS(=O)(=O)c1cc(C(=O)NC(CC2CC2)C2CCCN2)c2c(c1N)CCCO2

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 2/20 0.30
ADRA2C P18825 2/20 0.30
KCNH2 Q12809 2/20 0.30
HTR1A P08908 1/20 0.30
ACHE P22303 1/20 0.30
PTGS1 P23219 1/20 0.30
ADRA1A P35348 1/20 0.30
HTR3A P46098 1/20 0.30
LMNA P02545 1/20 0.30
ADRA2A P08913 1/20 0.30
DRD2 P14416 1/20 0.30
ALOX15 P16050 1/20 0.30
TSHR P16473 1/20 0.30
ADRA2B P18089 1/20 0.30
HTR2A P28223 1/20 0.30
MAPK1 P28482 1/20 0.30
HTR7 P34969 1/20 0.30
HRH1 P35367 1/20 0.30
DRD3 P35462 1/20 0.30
HTR2B P41595 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9869750 0.91 HTR4 (0.30) HTR4ADRA2CKCNH2HTR1AACHE
SCHEMBL9868594 0.91 BACE1 (0.30)
Hydrochloric Acid SCHEMBL9866623 0.90
SCHEMBL9822959 0.83 DRD2 (0.30) DRD2
SCHEMBL9868848 0.83 BACE1 (0.33) TSHR
Hydrochloric Acid SCHEMBL9868759 0.82 BACE1 (0.31)
SCHEMBL9823201 0.78
SCHEMBL10559503 0.77 DRD2 (0.53) HTR4ADRA2CKCNH2ACHEPTGS1
SCHEMBL27376806 0.77 ADRA2C (0.31) HTR4ADRA2CKCNH2HTR1AACHE
SCHEMBL10564984 0.75 DRD2 (0.52) HTR4ADRA2CKCNH2ACHEPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5006570-A Dihydrobenzofuran- and chroman-carboxamide derivatives, processes for the preparation thereof and use thereof as neuroleptics LABORATOIRES DELAGRANGE (FR) 1991-04-09 US disclosed