SCHEMBL9869982

SCHEMBL9869982

CCOC(=O)c1nc(COC)c(CC)c(COC)c1C(=O)OCC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 4/20 0.42
GABRA1 P14867 4/20 0.39
GABRA5 P31644 4/20 0.39
GABRA3 P34903 4/20 0.39
GABRA2 P47869 4/20 0.39
GABRA6 Q16445 4/20 0.39
GABRP O00591 3/20 0.39
GABRD O14764 3/20 0.39
GABRB1 P18505 3/20 0.39
GABRG2 P18507 3/20 0.39
GABRB3 P28472 3/20 0.39
GABRB2 P47870 3/20 0.39
GABRA4 P48169 3/20 0.39
GABRE P78334 3/20 0.39
GABRG1 Q8N1C3 3/20 0.39
GABRG3 Q99928 3/20 0.39
GABRQ Q9UN88 3/20 0.39
CYP1A2 P05177 2/20 0.38
CYP2C19 P33261 1/20 0.38
NR1H2 P55055 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9868508 0.75 GABRA1 (0.49) GABRA1GABRA5GABRA3GABRA2GABRA6
SCHEMBL9869186 0.71 CA12 (0.42) CYP1A2NR1H2NR1H3ALDH1A1HPGD
SCHEMBL9869495 0.71 CA12 (0.42) ALDH1A1HPGDCYP3A4GAA
SCHEMBL9868657 0.70 NR1H2 (0.44) GABRA1GABRA5GABRA3GABRA2GABRA6
SCHEMBL16851079 0.69 ADORA3 (0.65) ADORA3CYP1A2CYP2C19PDE4DALDH1A1
SCHEMBL9785613 0.68 NR1H2 (0.44) CYP1A2CYP2C19NR1H2NR1H3PDE4D
SCHEMBL8832474 0.67 ADORA3 (0.42) ADORA3CYP1A2CYP2C19ALDH1A1HPGD
SCHEMBL9868685 0.66 BRD4 (0.46) GABRA1GABRA5GABRA3GABRA2GABRA6
SCHEMBL25238862 0.66 PDE4D (0.49) NR1H2NR1H3PDE4DALDH1A1HPGD
SCHEMBL20135721 0.66 CA12 (0.44) GABRA1GABRA5GABRA3GABRA2GABRA6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997947-A Forming 6-substituted pyridine-2,3-dicarboxylic esters followed by reacting with aminoalkanecarboxylic acid amide; herbicides, plant growth regulators CIBA-GEIGY CORPORATION (US) 1991-03-05 US disclosed