SCHEMBL9870239

SCHEMBL9870239

Cc1cc(-c2cccc(C(F)(F)F)c2)n2ccnc2n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.43
ALDH1A1 P00352 1/20 0.43
GAA P10253 2/20 0.42
MAPT P10636 1/20 0.42
KMO O15229 1/20 0.41
HSD17B10 Q99714 2/20 0.41
KMT2A Q03164 1/20 0.41
CYP17A1 P05093 1/20 0.41
DYRK1A Q13627 4/20 0.41
DYRK2 Q92630 4/20 0.41
CCNA2 P20248 3/20 0.40
CDK2 P24941 3/20 0.40
CDK5 Q00535 3/20 0.40
CDK5R1 Q15078 3/20 0.40
DYRK1B Q9Y463 3/20 0.40
DYRK3 O43781 2/20 0.40
CCNT1 O60563 2/20 0.40
CDK9 P50750 2/20 0.40
LMNA P02545 1/20 0.40
PDE2A O00408 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9870207 0.82 KDM4E (0.49) KDM4EALDH1A1GAAMAPTKMO
SCHEMBL9870091 0.81 KDM4E (0.55) KDM4EALDH1A1GAAMAPTHSD17B10
SCHEMBL11009952 0.77 CYP2A6 (0.46) KDM4EALDH1A1MAPTKMT2A
SCHEMBL11009148 0.75 BACE1 (0.49) KDM4EALDH1A1MAPTHSD17B10DYRK1A
SCHEMBL5259449 0.75 BACE1 (0.64) KDM4EALDH1A1GAAMAPTCYP17A1
SCHEMBL9534839 0.74 HSD17B10 (0.49) KDM4EALDH1A1HSD17B10KMT2ADYRK1A
SCHEMBL9869878 0.73 KDM4E (0.44) KDM4EALDH1A1GAAMAPTKMO
SCHEMBL11467433 0.73 KDM4E (0.54) KDM4EALDH1A1GAAMAPTKMO
SCHEMBL5262408 0.73 GABRA1 (0.64)
SCHEMBL11463603 0.72 KDM4E (0.46) KDM4EALDH1A1HSD17B10CYP17A1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5037980-A Anxiolytic agents, hypotensive agents AMERICAN CYANAMID COMPANY (US) 1991-08-06 US claimed
US-5037980-A Anxiolytic agents, hypotensive agents AMERICAN CYANAMID COMPANY (US) 1991-08-06 US disclosed