SCHEMBL9870091

SCHEMBL9870091

Cc1cc(-c2ccccc2)n2ccnc2n1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.55
MAPT P10636 4/20 0.55
MAPK1 P28482 2/20 0.55
ALDH1A1 P00352 5/20 0.48
HPGD P15428 4/20 0.48
HSD17B10 Q99714 3/20 0.48
CHEK1 O14757 1/20 0.46
MAP4K4 O95819 1/20 0.46
CSF1R P07333 1/20 0.46
PRKACA P17612 1/20 0.46
KDR P35968 1/20 0.46
CDK8 P49336 1/20 0.46
MAP2K1 Q02750 1/20 0.46
ACVR1 Q04771 1/20 0.46
MAP4K2 Q12851 1/20 0.46
ROCK1 Q13464 1/20 0.46
DYRK1A Q13627 1/20 0.46
AURKB Q96GD4 1/20 0.46
DYRK1B Q9Y463 1/20 0.46
ADORA2A P29274 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11009148 0.87 BACE1 (0.49) KDM4EMAPTMAPK1ALDH1A1HPGD
SCHEMBL11009952 0.86 CYP2A6 (0.46) KDM4EMAPTMAPK1ALDH1A1KDR
SCHEMBL9870239 0.81 KDM4E (0.43) KDM4EMAPTALDH1A1HSD17B10DYRK1A
SCHEMBL9869878 0.79 KDM4E (0.44) KDM4EMAPTMAPK1ALDH1A1HPGD
SCHEMBL9870867 0.79 GABRA1 (0.42) KDM4EMAPTMAPK1CDK8MAP2K1
SCHEMBL9869785 0.75 TUBB4A (0.45) KDM4EMAPTALDH1A1HPGDSMN1; SMN2
SCHEMBL259043 0.73 KDM4E (0.50) KDM4EMAPTALDH1A1HPGDHSD17B10
SCHEMBL12395111 0.71 PDE2A (0.38) KDM4EMAPK1ALDH1A1HPGDADORA2A
SCHEMBL1681613 0.70 PDE2A (0.40) KDM4EALDH1A1HPGDHSD17B10MAP2K1
SCHEMBL1681759 0.70 DPP4 (0.39) KDM4EALDH1A1HPGDMAP2K1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5037980-A Anxiolytic agents, hypotensive agents AMERICAN CYANAMID COMPANY (US) 1991-08-06 US disclosed