SCHEMBL9869878

SCHEMBL9869878

Cc1cc(-c2ccc(Cl)c(Cl)c2)n2ccnc2n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.44
ALDH1A1 P00352 5/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
HPGD P15428 3/20 0.44
NPC1 O15118 2/20 0.44
MAPT P10636 2/20 0.44
RAB9A P51151 2/20 0.44
EGLN2 Q96KS0 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
MEN1 O00255 1/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
KMT2A Q03164 1/20 0.40
RELA Q04206 1/20 0.40
HSD17B10 Q99714 2/20 0.38
MAPK1 P28482 1/20 0.38
TSHR P16473 1/20 0.38
DPP4 P27487 1/20 0.38
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9870091 0.79 KDM4E (0.55) KDM4EALDH1A1SMN1; SMN2HPGDNPC1
SCHEMBL11009148 0.79 BACE1 (0.49) KDM4EALDH1A1SMN1; SMN2HPGDMAPT
SCHEMBL11009952 0.75 CYP2A6 (0.46) KDM4EALDH1A1SMN1; SMN2MAPTKMT2A
SCHEMBL9870239 0.73 KDM4E (0.43) KDM4EALDH1A1MAPTKMT2AHSD17B10
SCHEMBL1681759 0.73 DPP4 (0.39) KDM4EALDH1A1SMN1; SMN2HPGDRAB9A
SCHEMBL9869785 0.70 TUBB4A (0.45) KDM4EALDH1A1SMN1; SMN2HPGDMAPT
SCHEMBL9329531 0.70 PDE2A (0.37) KDM4EALDH1A1HPGDNPC1RAB9A
SCHEMBL259043 0.69 KDM4E (0.50) KDM4EALDH1A1SMN1; SMN2HPGDNPC1
SCHEMBL9870867 0.69 GABRA1 (0.42) KDM4EMAPTMAPK1PDE2A
SCHEMBL10562568 0.67 HSD11B1 (0.46) KDM4EALDH1A1SMN1; SMN2HPGDNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5037980-A Anxiolytic agents, hypotensive agents AMERICAN CYANAMID COMPANY (US) 1991-08-06 US claimed
US-5037980-A Anxiolytic agents, hypotensive agents AMERICAN CYANAMID COMPANY (US) 1991-08-06 US disclosed