SCHEMBL9870279

SCHEMBL9870279

CC1=C(c2cccc(Cl)c2)n2ncc(C(N)=O)c2NC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.40
PARP1 P09874 1/20 0.40
TLR8 Q9NR97 2/20 0.38
IKBKB O14920 2/20 0.38
CHUK O15111 1/20 0.38
JAK2 O60674 6/20 0.38
JAK1 P23458 2/20 0.38
TYK2 P29597 2/20 0.38
JAK3 P52333 2/20 0.38
KCNH2 Q12809 1/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
ATM Q13315 1/20 0.38
KMT2A Q03164 1/20 0.37
NUDT1 P36639 1/20 0.36
FGFR1 P11362 1/20 0.36
FGFR2 P21802 1/20 0.36
FGFR3 P22607 1/20 0.36
IKBKE Q14164 1/20 0.35
PIN1 Q13526 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9868786 0.86 TSHR (0.39) PARP1IKBKBCHUKJAK2JAK1
SCHEMBL9869743 0.84 KDM4E (0.50) PARP1IKBKBJAK2NPC1RAB9A
SCHEMBL9478335 0.78 RXRA (0.46) NPC1RAB9AATMKMT2ANUDT1
SCHEMBL8337977 0.69 TLR8 (0.50) PARP1TLR8JAK2JAK1TYK2
SCHEMBL2834342 0.66 RIPK2 (0.70) HTTPARP1NPC1RAB9AATM
SCHEMBL8335601 0.65 RIPK2 (0.46) JAK2JAK1TYK2JAK3NPC1
SCHEMBL8339312 0.65 CDC7 (0.43) JAK2JAK1TYK2JAK3KCNH2
SCHEMBL30927156 0.64 MKNK1 (0.60) PARP1IKBKBCHUKJAK2NPC1
SCHEMBL15428638 0.63 DCAF1 (0.54) PARP1IKBKBCHUKJAK2JAK1
SCHEMBL27922044 0.62 PARP1 (0.55) PARP1IKBKBCHUKJAK2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5013737-A Hypotensive, anxiolytic, cognitive disorders AMERICAN CYANAMID COMPANY (US) 1991-05-07 US disclosed