SCHEMBL9870480

SCHEMBL9870480

CNCc1cccc(CSCCN)c1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.46
CYP2D6 P10635 2/20 0.46
CYP2C19 P33261 2/20 0.46
NOS1 P29475 4/20 0.44
PRMT6 Q96LA8 7/20 0.41
CYP3A4 P08684 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MAPT P10636 1/20 0.41
EPHX2 P34913 1/20 0.40
NOS3 P29474 2/20 0.38
HTR7 P34969 1/20 0.38
CYP2C9 P11712 1/20 0.38
KIF11 P52732 1/20 0.36
NOS2 P35228 1/20 0.36
TP53 P04637 1/20 0.36
SLC11A2 P49281 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dimethylamine SCHEMBL9872444 0.80 TAAR1 (0.53) CYP1A2CYP2D6CYP2C19CYP3A4KDM4E
SCHEMBL1697126 0.78 MAPT (0.64) NOS1PRMT6CYP3A4KDM4EMAPT
SCHEMBL15022828 0.77 TAAR1 (0.58) CYP1A2CYP2D6CYP2C19CYP3A4KDM4E
SCHEMBL9872439 0.77 ACHE (0.53) CYP1A2CYP2D6CYP2C19NOS1PRMT6
SCHEMBL3363042 0.76 NOS1 (0.53) NOS1PRMT6CYP3A4KDM4EMAPT
SCHEMBL30125422 0.76 NOS1 (0.53) NOS1PRMT6CYP3A4KDM4EMAPT
Hydrochloric Acid SCHEMBL10955274 0.75 ACHE (0.51) CYP1A2CYP2D6CYP2C19NOS1PRMT6
Hydrochloric Acid SCHEMBL3273205 0.75 MAPT (0.68) NOS1PRMT6CYP3A4KDM4EMAPT
SCHEMBL11745386 0.74 TAAR1 (0.58) CYP1A2CYP2D6CYP2C19KIF11TP53
SCHEMBL15023253 0.74 IDO1 (0.47) CYP1A2CYP2D6CYP2C19CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5021429-A Histamine h2-antagonists; antisecretory-antiallergen agent; skin disorders and peptic ulcers ALLEN & HANSBURYS LIMITED (GB) 1991-06-04 US disclosed
US-4496567-A HSITAMINE H2 ANTAGONISTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1985-01-29 US disclosed
EP-0013071-A1 Pyrimidinone derivatives, processes for preparing them and pharmaceutical compositions containing them SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1980-07-09 EP disclosed
WO-1980000966-A1 NEW HISTAMINE H2-ANTAGONISTS SMITH KLINE FRENCH LAB (GB) 1980-05-15 WO disclosed