SCHEMBL9870975

SCHEMBL9870975

Cc1ccc(S(=O)(=O)OC2=C(C(=O)OCc3ccc([N+](=O)[O-])cc3)N3C(=O)CC3C2)cc1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
MAPT P10636 1/20 0.49
HPGD P15428 1/20 0.49
NPC1 O15118 1/20 0.46
KMT2A Q03164 1/20 0.46
PLCG1 P19174 1/20 0.42
POLB P06746 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
ATM Q13315 1/20 0.39
ELANE P08246 1/20 0.39
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9871240 0.91 TDP1 (0.47) ALDH1A1PLCG1TDP1ATMELANE
SCHEMBL10570187 0.88 ELANE (0.51) MAPTHPGDELANE
SCHEMBL9824372 0.83 ALDH1A1 (0.43) ALDH1A1MAPTHPGDNPC1KMT2A
SCHEMBL10664044 0.83 ALDH1A1 (0.43) ALDH1A1MAPTHPGDNPC1KMT2A
SCHEMBL11066637 0.82 PLCG1 (0.53) ALDH1A1MAPTHPGDNPC1KMT2A
SCHEMBL9870805 0.78 ELANE (0.48) MAPTHPGDELANE
SCHEMBL9872583 0.77 CA1 (0.39) ALDH1A1KMT2ASMN1; SMN2
SCHEMBL11150895 0.77 RAB9A (0.47) ALDH1A1MAPTHPGDNPC1KMT2A
SCHEMBL9666113 0.76 ALDH1A1 (0.45) ALDH1A1MAPTHPGDNPC1KMT2A
SCHEMBL11148244 0.76 ALDH1A1 (0.44) ALDH1A1MAPTHPGDNPC1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5021566-A Carbapenicillins; preservatives; antiseptics; grampositive and gram negative bacteria MERCK & CO. INC. (US) 1991-06-04 US disclosed
US-4820817-A Process for preparing 3-substituted-6-substituted-7-oxo-1-azabicycl(3.2.0)-hept-2-ene-2-carboxylic acid MERCK & CO., INC. (US) 1989-04-11 US disclosed
US-4745188-A ANTIBIOTICS, SULFIDING MERCK & CO., INC. (US) 1988-05-17 US disclosed
US-4530841-A Antibiotic containing hetero ring MERCK & CO., INC. (US) 1985-07-23 US disclosed
US-4369187-A AMINO ACID DERIVATIVE ANTIBIOTICS MERCK & CO., INC. (US) 1983-01-18 US disclosed
US-4357342-A 1-Azabicyclo[3.2.0]heptan-3,7-dione-2-carboxylic acid MERCK & CO., INC. (US) 1982-11-02 US disclosed
US-4318912-A 6-(1-Hydroxyethyl)-3-substituted-1-azabicyclo(3.2.0)-hept-2-en-7-one-2-carboxylic acid MERCK & CO., INC. (US) 1982-03-09 US disclosed
US-4310538-A BACTERICIDES MERCK & CO., INC. (US) 1982-01-12 US disclosed