SCHEMBL9871979

SCHEMBL9871979

[N-]=[N+]=C(C(=O)CC1CC(=O)N1)C(=O)OCc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.41
ATM Q13315 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
RAB9A P51151 1/20 0.38
POLB P06746 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
IDO1 P14902 1/20 0.36
HTT P42858 1/20 0.36
HTR2A P28223 1/20 0.36
AKR1C3 P42330 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9871413 0.85 BRD4 (0.40) ALDH1A1RAB9ASMN1; SMN2
SCHEMBL10759407 0.79 RAB9A (0.35) TDP1ATMALDH1A1RAB9APOLB
SCHEMBL2944429 0.79 RAB9A (0.35) TDP1ATMRAB9APOLBSMN1; SMN2
SCHEMBL9168542 0.79 RAB9A (0.35) TDP1ATMRAB9APOLBSMN1; SMN2
SCHEMBL10790770 0.79 RAB9A (0.35) TDP1ATMRAB9APOLBSMN1; SMN2
SCHEMBL10493918 0.79 ALDH1A1 (0.37) ALDH1A1MAPTHPGDRAB9APOLB
SCHEMBL9670137 0.79 ALDH1A1 (0.39) TDP1ALDH1A1MAPTHPGDRAB9A
SCHEMBL9705614 0.79 TDP1 (0.39) TDP1ATMALDH1A1MAPTHPGD
SCHEMBL7186704 0.79 TDP1 (0.39) TDP1ATMALDH1A1MAPTHPGD
SCHEMBL10346269 0.78 HTR2A (0.39) ALDH1A1MAPTHPGDRAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5021566-A Carbapenicillins; preservatives; antiseptics; grampositive and gram negative bacteria MERCK & CO. INC. (US) 1991-06-04 US disclosed
US-4841042-A Process for the preparation of carbapenem intermediates BAYER AKTIENGESELLSCHAFT (DE) 1989-06-20 US disclosed
US-4820817-A Process for preparing 3-substituted-6-substituted-7-oxo-1-azabicycl(3.2.0)-hept-2-ene-2-carboxylic acid MERCK & CO., INC. (US) 1989-04-11 US disclosed
US-4745188-A ANTIBIOTICS, SULFIDING MERCK & CO., INC. (US) 1988-05-17 US disclosed
US-4707547-A AMINATION TO FORM ANTIBIOTIC MERCK & CO., INC. (US) 1987-11-17 US disclosed
EP-0195963-A1 Process for the preparation of carbapenem intermediates BAYER AG (DE) 1986-10-01 EP disclosed
US-4530841-A Antibiotic containing hetero ring MERCK & CO., INC. (US) 1985-07-23 US disclosed
EP-0134301-A1 6-(1'-Hydroxyethyl)-3-substituted amino-1-azabicyclo(3.2.0)-hept-2-en-7-one-2-carboxylic acid MERCK & CO. INC. (US) 1985-03-20 EP disclosed
US-4369187-A AMINO ACID DERIVATIVE ANTIBIOTICS MERCK & CO., INC. (US) 1983-01-18 US disclosed
US-4357342-A 1-Azabicyclo[3.2.0]heptan-3,7-dione-2-carboxylic acid MERCK & CO., INC. (US) 1982-11-02 US disclosed
US-4318912-A 6-(1-Hydroxyethyl)-3-substituted-1-azabicyclo(3.2.0)-hept-2-en-7-one-2-carboxylic acid MERCK & CO., INC. (US) 1982-03-09 US disclosed
US-4310538-A BACTERICIDES MERCK & CO., INC. (US) 1982-01-12 US disclosed