SCHEMBL9872861

SCHEMBL9872861

NC1(CCc2ccccc2)N=NN=N1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 9/20 0.45
MAOA P21397 8/20 0.45
KDM1A O60341 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
CYP2A6 P11509 1/20 0.43
HTR2A P28223 1/20 0.43
TAAR1 Q96RJ0 1/20 0.43
LOXL2 Q9Y4K0 1/20 0.43
ALDH1A1 P00352 2/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
ALOX12 P18054 1/20 0.39
CASP1 P29466 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CYP2D6 P10635 2/20 0.39
ATM Q13315 1/20 0.39
KEAP1 Q14145 1/20 0.39
NPC1 O15118 1/20 0.39
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9873163 0.78 MAOB (0.50) MAOBMAOAKDM1ASMN1; SMN2CYP2A6
SCHEMBL5247853 0.72 TDP1 (0.45) MAOBMAOAKDM1ASMN1; SMN2CYP2A6
SCHEMBL27639939 0.71 KDM1A (0.38) MAOBMAOAKDM1ASMN1; SMN2CYP2A6
SCHEMBL21058245 0.67 MAOA (0.52) MAOBMAOAKDM1ASMN1; SMN2CYP2A6
Hydrazine SCHEMBL4517324 0.66 MAOA (0.68) MAOBMAOAKDM1ASMN1; SMN2CYP2A6
Hydrochloric Acid SCHEMBL3787328 0.66 MAOB (0.65) MAOBMAOASMN1; SMN2CYP2A6HTR2A
SCHEMBL21058274 0.65 MAOA (0.50) MAOBMAOAKDM1ASMN1; SMN2CYP2A6
SCHEMBL28720281 0.65 KDM1A (0.47) MAOBMAOAKDM1ASMN1; SMN2CYP2A6
SCHEMBL21058226 0.65 MAOA (0.43) MAOBMAOAKDM1ASMN1; SMN2CYP2A6
SCHEMBL28282400 0.65 KDM1A (0.47) MAOBMAOAKDM1ASMN1; SMN2CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991017150-A1 TETRAZOLE UREA AND THIOUREA ACAT INHIBITORS WARNER-LAMBERT COMPANY (US) 1991-11-14 WO disclosed