SCHEMBL9872863

SCHEMBL9872863

COc1cc(N)c(Cl)cc1C(=O)OC1CC2CCC(C1)N2Cc1ccccc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.67
HTR4 Q13639 1/20 0.56
DRD4 P21917 6/20 0.55
DRD3 P35462 4/20 0.55
ACHE P22303 2/20 0.55
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
ADRA2A P08913 1/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C9 P11712 1/20 0.55
ADRA2B P18089 1/20 0.55
ADRA2C P18825 1/20 0.55
SLC6A2 P23975 1/20 0.55
HTR2A P28223 1/20 0.55
HTR2C P28335 1/20 0.55
ADRA1A P35348 1/20 0.55
OPRK1 P41145 1/20 0.55
HTR2B P41595 1/20 0.55
CHRNA4 P43681 1/20 0.55
HTR3A P46098 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9872858 1.00 DRD2 (0.67) DRD2HTR4DRD4DRD3ACHE
SCHEMBL9872901 0.82 POLB (0.49) DRD2DRD4DRD3KCNH2
SCHEMBL9872897 0.82 POLB (0.49) DRD2DRD4DRD3KCNH2
SCHEMBL9872909 0.81 DRD2 (0.46) DRD2DRD4DRD3OPRK1HTR3A
SCHEMBL11094874 0.78 DRD2 (0.61) DRD2DRD4DRD3ACHECYP1A2
SCHEMBL11093546 0.77 DRD2 (0.60) DRD2DRD4DRD3ACHECYP1A2
SCHEMBL7444398 0.76 HTR4 (0.55) HTR4CYP3A4
SCHEMBL7444394 0.76 HTR4 (0.55) HTR4CYP3A4
SCHEMBL11237006 0.76 DRD2 (0.83) DRD2HTR4DRD4DRD3ACHE
SCHEMBL11228982 0.76 DRD2 (0.83) DRD2HTR4DRD4DRD3ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5017582-A Analgesics SANDOZ LTD. (CH) 1991-05-21 US disclosed
US-4910207-A Antipsychotic agent NOVARTIS AG (CH) 1990-03-20 US disclosed
US-4803199-A SEROTONIN ANTAGONIST, ANALGESIC ANTIARRHYTHMIC AGENTS NOVARTIS AG (CH) 1989-02-07 US disclosed