SCHEMBL9876492

SCHEMBL9876492

COC(=O)c1ccc(C#Cc2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.55
LMNA P02545 1/20 0.52
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
NOTUM Q6P988 2/20 0.47
RARB P10826 1/20 0.47
RARG P13631 1/20 0.47
MAPT P10636 2/20 0.47
CA1 P00915 2/20 0.47
CA2 P00918 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
CA12 O43570 1/20 0.47
CA7 P43166 1/20 0.47
CA9 Q16790 1/20 0.47
CA14 Q9ULX7 1/20 0.47
CFTR P13569 1/20 0.46
P2RY6 Q15077 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL385370 0.89 LMNA (0.60) LMNACES2CES1NOTUMMAPT
Ammonia Solution, Strong SCHEMBL27316369 0.88 LMNA (0.59) LMNACES2CES1NOTUMMAPT
SCHEMBL69268 0.86 PTPN11 (0.69) PTPN11MAPTCA1CA2TDP1
SCHEMBL29893239 0.85 CFTR (0.50) PTPN11LMNANOTUMMAPTCFTR
SCHEMBL13063663 0.84 LMNA (0.56) LMNACES2CES1NOTUMMAPT
SCHEMBL2271347 0.84 LMNA (0.56) LMNACES2CES1NOTUMMAPT
SCHEMBL22096409 0.84 CA12 (0.50) PTPN11LMNANOTUMCA1CA2
SCHEMBL31710343 0.84 CFTR (0.56) PTPN11LMNANOTUMMAPTCFTR
SCHEMBL31575935 0.83 SRD5A2 (0.65) LMNACES2CES1NOTUMMAPT
Methylene Chloride SCHEMBL28147089 0.83 LMNA (0.55) LMNACES2CES1NOTUMMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0407955-A1 New hetrazepines acting as PAF antagonists, process for their production and their use as drugs BOEHRINGER INGELHEIM KG (DE) 1991-01-16 EP disclosed