SCHEMBL9876593

SCHEMBL9876593

[c]1ccc2ccccc2n1.[c]1ncccn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.41
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.37
MAPT P10636 2/20 0.37
GLA P06280 1/20 0.37
ACHE P22303 1/20 0.37
NCF1 P14598 3/20 0.36
NOS2 P35228 1/20 0.36
BACE1 P56817 1/20 0.36
CA12 O43570 1/20 0.36
CA9 Q16790 1/20 0.36
RAB9A P51151 4/20 0.35
NPC1 O15118 3/20 0.35
CYP3A4 P08684 1/20 0.35
AR P10275 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
KDM4E B2RXH2 2/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2910 0.88 CYP1A2 (0.44) CYP1A2ALDH1A1HPGDMAPTGLA
SCHEMBL7374426 0.73 CYP1A2 (0.33) CYP1A2ALDH1A1
SCHEMBL20659316 0.71 MAPT (0.54) CYP1A2ALDH1A1HPGDMAPTGLA
SCHEMBL524746 0.69 ALDH1A1 (0.46) CYP1A2ALDH1A1HPGDMAPTGLA
SCHEMBL2139252 0.68 ALDH1A1 (0.44) CYP1A2ALDH1A1HPGDMAPTGLA
SCHEMBL16357 0.65 KDM4E (0.32) CYP1A2ALDH1A1CYP3A4CYP2D6CYP2C9
SCHEMBL16316 0.65 MAP4K4 (0.34)
SCHEMBL2671574 0.65 NPC1 (0.47) CYP1A2ALDH1A1MAPTRAB9ANPC1
SCHEMBL3032 0.64 ALDH1A1 (0.44) CYP1A2ALDH1A1HPGDMAPTGLA
SCHEMBL449631 0.64

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0156433-B1 ANTI-VIRALLY ACTIVE PYRIDAZINAMINES JANSSEN PHARMACEUTICA N.V. (BE) 1991-02-27 EP claimed
EP-0156433-B1 ANTI-VIRALLY ACTIVE PYRIDAZINAMINES JANSSEN PHARMACEUTICA N.V. (BE) 1991-02-27 EP disclosed