SCHEMBL9879719

SCHEMBL9879719

CN(C)CCCOc1ccc(N2N=C3c4cc(OCCCN(C)C)ccc4CCC3CC2=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.43
MAPK14 Q16539 1/20 0.41
HRH3 Q9Y5N1 3/20 0.40
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
ESR1 P03372 1/20 0.37
THRA P10827 1/20 0.37
THRB P10828 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
DRD2 P14416 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9601499 0.93 ACHE (0.41) ACHEMAPK14HRH3CYP1A2CYP3A4
Maleic Acid SCHEMBL9865891 0.90 ACHE (0.38) ACHEMAPK14HRH3THRBMEN1
Fumaric Acid SCHEMBL9865899 0.90 ACHE (0.38) ACHEMAPK14HRH3THRBMEN1
SCHEMBL9601994 0.86 ACHE (0.40) ACHEHRH3DRD2
Water SCHEMBL9865858 0.85 HRH3 (0.37) HRH3DRD2
Water SCHEMBL9865856 0.85 HRH3 (0.37) HRH3DRD2
Fumaric Acid SCHEMBL9868348 0.82 L3MBTL1 (0.37) ACHEMAPK14HRH3THRBMEN1
Fumaric Acid SCHEMBL9601552 0.82 L3MBTL1 (0.37) ACHEMAPK14HRH3THRBMEN1
SCHEMBL9865917 0.81 MAOA (0.34) ACHEHRH3MEN1KMT2A
SCHEMBL9867304 0.81 MAOA (0.35) ACHEHRH3MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5045541-A Immunodeficiency disorders YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1991-09-03 US disclosed
EP-0351435-A1 FUSED PYRIDAZINE COMPOUNDS AND THEIR MEDICINAL USES Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1990-01-24 EP disclosed