SCHEMBL988730

SCHEMBL988730

O=C([O-])CC(O)(C(=O)[O-])C(O)C(=O)[O-].[Cr+3]

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CA4 P22748 3/20 0.43
CPT2 P23786 1/20 0.33
ACLY P53396 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL990294 1.00 CA4 (0.43) CA4CPT2ACLY
SCHEMBL30463175 0.96 CA4 (0.43) CA4CPT2ACLY
SCHEMBL965645 0.96 CA4 (0.48) CA4CPT2ACLY
SCHEMBL336805 0.96 CA4 (0.43) CA4CPT2ACLY
SCHEMBL966173 0.96 CA4 (0.43) CA4CPT2ACLY
SCHEMBL31473016 0.96 CA4 (0.48) CA4CPT2ACLY
SCHEMBL1460547 0.96 CA4 (0.43) CA4CPT2ACLY
Potassium Ion SCHEMBL337213 0.96 CA4 (0.43) CA4CPT2ACLY
Zinc Ion SCHEMBL2315207 0.96 CA4 (0.43) CA4CPT2ACLY
SCHEMBL2487788 0.96 CA4 (0.43) CA4CPT2ACLY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4070801-A1 COMPOSITIONS OF INSULIN AND CHROMIUM FOR THE TREATMENT AND PREVENTION OF DIABETES, HYPOGLYCEMIA AND RELATED DISORDERS Nutrition 21, LLC (US) 2022-10-12 EP disclosed
EP-3513790-A1 CHROMIUM COMPLEXES AS ENHANCERS OF BRAIN GLUCOSE TRANSPORTERS JDS Therapeutics, LLC (US) 2019-07-24 EP disclosed
EP-2448412-B1 CHROMIUM COMPLEXES AS ENHANCERS OF BRAIN GLUCOSE TRANSPORTERS JDS THERAPEUTICS LLC (US) 2019-05-01 EP disclosed
US-9700546-B2 Trivalent chromium compounds, compositions and methods of use INTERHEALTH NUTRACEUTICALS, INC. (US) 2017-07-11 US disclosed
US-20160354353-A9 TRIVALENT CHROMIUM COMPOUNDS, COMPOSITIONS AND METHODS OF USE LONZA CONSUMER HEALTH INC. 2016-12-08 US disclosed
US-20160220581-A1 CHROMIUM COMPOSITIONS FOR THE TREATMENT OR PREVENTION OF DIABETIC RETINOPATHY CAPITAL ONE, NATIONAL ASSOCIATION, AS AGENT 2016-08-04 US disclosed
US-20150306083-A1 TRIVALENT CHROMIUM COMPOUNDS, COMPOSITIONS AND METHODS OF USE INTERHEALTH NUTRACEUTICALS INC (US) 2015-10-29 US disclosed
US-20150224140-A1 CHROMIUM COMPLEXES AS ENHANCERS OF BRAIN GLUCOSE TRANSPORTERS CAPITAL ONE, NATIONAL ASSOCIATION, AS AGENT 2015-08-13 US disclosed
US-9028879-B2 Chromium complexes as enhancers of brain glucose transporters JDS THERAPEUTICS, LLC (US) 2015-05-12 US disclosed
US-20150094258-A1 METHODS AND COMPOSITIONS FOR THE TREATMENT AND PREVENTION OF HYPOGLYCEMIA AND RELATED DISORDERS JDS THERAPEUTICS LLC (US) 2015-04-02 US disclosed
US-8933022-B2 Methods and compositions for the treatment and prevention Hypoglycemia and related disorders JDS THERAPEUTICS, LLC (US) 2015-01-13 US disclosed
WO-2012119007-A1 COMPOSITIONS OF INSULIN AND CHROMIUM FOR THE TREATMENT AND PREVENTION OF DIABETES, HYPOGLYCEMIA AND RELATED DISORDERS N21 ACQUISITION HOLDING, LLC (US) 2012-09-07 WO disclosed
US-20120225134-A1 METHODS AND COMPOSITIONS FOR THE TREATMENT AND PREVENTION OF HYPOGLYCEMIA AND RELATED DISORDERS N21 ACQUISITION HOLDING, LLC (US) 2012-09-06 US disclosed
EP-2448412-A1 CHROMIUM COMPLEXES AS ENHANCERS OF BRAIN GLUCOSE TRANSPORTERS Nutrition 21, Inc. (US) 2012-05-09 EP disclosed
US-20120100228-A1 CHROMIUM COMPLEXES AS ENHANCERS OF BRAIN GLUCOSE TRANSPORTERS CAPITAL ONE, NATIONAL ASSOCIATION, AS AGENT 2012-04-26 US disclosed
WO-2011002939-A1 CHROMIUM COMPLEXES AS ENHANCERS OF BRAIN GLUCOSE TRANSPORTERS NUTRITION 21, INC. (US) 2011-01-06 WO disclosed
US-20090092560-A1 TRIVALENT CHROMIUM COMPOUNDS, COMPOSITIONS AND METHODS OF USE INTERHEALTH NUTRACEUTICALS, INC. (US) 2009-04-09 US disclosed
EP-2012770-A2 TRIVALENT CHROMIUM COMPOUNDS, COMPOSITIONS AND METHODS OF USE Interhealth Nutraceuticals, Inc. (US) 2009-01-14 EP disclosed
WO-2007121312-A9 TRIVALENT CHROMIUM COMPOUNDS, COMPOSITIONS AND METHODS OF USE INTERHEALTH NUTRACEUTICALS INC (US) 2008-07-17 WO disclosed
WO-2007121312-A2 TRIVALENT CHROMIUM COMPOUNDS, COMPOSITIONS AND METHODS OF USE INTERHEALTH NUTRACEUTICALS, INC. (US) 2007-10-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120100228-A1 CHROMIUM COMPLEXES AS ENHANCERS OF BRAIN GLUCOSE TRANSPORTERS SLC2A3, SLC2A1, SLC2A2 CA4 680/4885CPT2 288/4885ACLY 230/4885
US-20150094258-A1 METHODS AND COMPOSITIONS FOR THE TREATMENT AND PREVENTION OF HYPOGLYCEMIA AND RELATED DISORDERS IAPP, GCG, PYGL CA4 95/4885CPT2 822/4885ACLY 258/4885
US-20160220581-A1 CHROMIUM COMPOSITIONS FOR THE TREATMENT OR PREVENTION OF DIABETIC RETINOPATHY RBP4, RBP1, ALDH1A2 CA4 169/4885CPT2 733/4885ACLY 904/4885
US-20150224140-A1 CHROMIUM COMPLEXES AS ENHANCERS OF BRAIN GLUCOSE TRANSPORTERS SLC2A3, SLC2A1, SLC2A2 CA4 680/4885CPT2 288/4885ACLY 230/4885
US-20120225134-A1 METHODS AND COMPOSITIONS FOR THE TREATMENT AND PREVENTION OF HYPOGLYCEMIA AND RELATED DISORDERS IAPP, GCG, PYGL CA4 95/4885CPT2 822/4885ACLY 258/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.