SCHEMBL988802

SCHEMBL988802

[c]1cccc(-c2cncnc2)n1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.41
CYP2A6 P11509 3/20 0.39
PIM1 P11309 1/20 0.32
CYP19A1 P11511 1/20 0.31
AXL P30530 1/20 0.31
PBRM1 Q86U86 1/20 0.31
MKNK1 Q9BUB5 1/20 0.31
MKNK2 Q9HBH9 1/20 0.31
ALDH1A1 P00352 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL988803 0.80 CYP2A6 (0.53) CYP2A6CYP19A1AXLPBRM1MKNK1
SCHEMBL1201737 0.77 LMNA (0.42) CYP19A1ALDH1A1CYP1A2CYP3A4
SCHEMBL16834631 0.76 CYP2A6 (0.41) CYP2A6PIM1CYP3A4
SCHEMBL1316597 0.76 RAB9A (0.48) ALDH1A1
SCHEMBL988804 0.73
SCHEMBL18422490 0.72 CYP11B2 (0.43)
SCHEMBL6544558 0.71 MAPT (0.54) CYP19A1MKNK1MKNK2ALDH1A1
SCHEMBL5541082 0.71 SREBF2 (0.41) ALDH1A1
SCHEMBL12614991 0.71 CYP1A2 (0.39) CYP19A1ALDH1A1CYP1A2
SCHEMBL11297134 0.71 GRM2 (0.37) ATMALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011008788-A1 FLUORO-SUBSTITUTED COMPOUNDS AS KINASE INHIBITORS AND METHODS OF USE THEREOF ZHANG DAWEI (US) 2011-01-20 WO claimed
WO-2011008788-A1 FLUORO-SUBSTITUTED COMPOUNDS AS KINASE INHIBITORS AND METHODS OF USE THEREOF ZHANG DAWEI (US) 2011-01-20 WO disclosed