SCHEMBL989371

SCHEMBL989371

CCOC(=O)c1cc2c(s1)CCOc1ccc(Br)cc1-2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.41
ALDH1A1 P00352 4/20 0.41
HPGD P15428 3/20 0.41
TDP1 Q9NUW8 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
NPC1 O15118 4/20 0.40
RAB9A P51151 4/20 0.40
CLK1 P49759 1/20 0.40
MAPT P10636 6/20 0.40
GLA P06280 1/20 0.40
GAA P10253 1/20 0.40
ATM Q13315 1/20 0.40
ALPL P05186 1/20 0.38
ALOX5 P09917 3/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
USP2 O75604 1/20 0.37
LMNA P02545 1/20 0.37
MAPK1 P28482 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL988662 0.85 ALDH1A1 (0.52) KDM4EALDH1A1HPGDTDP1L3MBTL1
SCHEMBL988679 0.83 KDM4E (0.57) KDM4EALDH1A1HPGDTDP1L3MBTL1
SCHEMBL988982 0.82 NOTUM (0.39) KDM4EALDH1A1HPGDNPC1RAB9A
SCHEMBL991392 0.81 NOTUM (0.50) NPC1RAB9AMAPTMEN1KMT2A
SCHEMBL989938 0.81 ALDH1A1 (0.41) KDM4EALDH1A1NPC1RAB9AGAA
SCHEMBL1484646 0.80 MAP3K14 (0.48) NPC1RAB9ACLK1OGA
SCHEMBL4055690 0.77 LMNA (0.36) KDM4EALDH1A1L3MBTL1NPC1RAB9A
SCHEMBL1484604 0.73 PIK3CA (0.42) NPC1RAB9ACLK1OGA
SCHEMBL1516838 0.72 SRD5A1 (0.38) KDM4EALDH1A1HPGDMAPTGAA
SCHEMBL16794102 0.72 KDM4E (0.44) KDM4EALDH1A1HPGDTDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2276767-A1 BENZOPYRAN AND BENZOXEPIN PI3K INHIBITOR COMPOUNDS AND METHODS OF USE Genentech, Inc. (US) 2011-01-26 EP disclosed
WO-2009123971-A1 BENZOPYRAN AND BENZOXEPIN PI3K INHIBITOR COMPOUNDS AND METHODS OF USE GENENTECH, INC. (US) 2009-10-08 WO disclosed