SCHEMBL989938

SCHEMBL989938

NNC(=O)c1cc2c(s1)CCOc1ccc(Br)cc1-2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
GAA P10253 3/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
LMNA P02545 1/20 0.38
CASP3 P42574 1/20 0.37
SENP8 Q96LD8 1/20 0.37
SENP7 Q9BQF6 1/20 0.37
SENP6 Q9GZR1 1/20 0.37
NOTUM Q6P988 1/20 0.37
RAB9A P51151 5/20 0.36
NPC1 O15118 4/20 0.36
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MAOB P27338 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL991392 0.86 NOTUM (0.50) MEN1KMT2ALMNANOTUMRAB9A
SCHEMBL988982 0.85 NOTUM (0.39) ALDH1A1MEN1KMT2AGAALMNA
SCHEMBL988065 0.81 THRB (0.42) ALDH1A1MEN1KMT2AGAACYP3A4
SCHEMBL989371 0.81 KDM4E (0.41) ALDH1A1MEN1KMT2AGAACYP1A2
SCHEMBL4055690 0.80 LMNA (0.36) ALDH1A1MEN1KMT2AGAALMNA
SCHEMBL1619624 0.78 MAP3K14 (0.50) PIK3CDPIK3R1MAP3K14
SCHEMBL988878 0.75 NOTUM (0.55) ALDH1A1MEN1KMT2AGAACYP1A2
SCHEMBL1516838 0.75 SRD5A1 (0.38) ALDH1A1GAALMNANOTUMMAOB
SCHEMBL989368 0.72 ALDH1A1 (0.38) ALDH1A1MEN1KMT2AGAACYP3A4
SCHEMBL988463 0.69 NOTUM (0.70) ALDH1A1GAANOTUMMAP3K14KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2276767-A1 BENZOPYRAN AND BENZOXEPIN PI3K INHIBITOR COMPOUNDS AND METHODS OF USE Genentech, Inc. (US) 2011-01-26 EP disclosed
WO-2009123971-A1 BENZOPYRAN AND BENZOXEPIN PI3K INHIBITOR COMPOUNDS AND METHODS OF USE GENENTECH, INC. (US) 2009-10-08 WO disclosed