SCHEMBL9899776

SCHEMBL9899776

OCCCC(c1ccccc1)c1ccccc1Br

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.42
TDO2 P48775 1/20 0.42
HRH1 P35367 4/20 0.41
HTR2A P28223 4/20 0.41
ALDH1A1 P00352 2/20 0.40
CYP3A4 P08684 1/20 0.40
ALOX15 P16050 1/20 0.40
CYP2C19 P33261 1/20 0.40
OPRM1 P35372 2/20 0.36
OPRD1 P41143 2/20 0.36
OPRK1 P41145 2/20 0.36
OPRL1 P41146 2/20 0.36
TRPA1 O75762 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
LMNA P02545 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CYP19A1 P11511 2/20 0.35
HTT P42858 1/20 0.34
GRM2 Q14416 1/20 0.34
GRM3 Q14832 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9899643 0.81 TBXAS1 (0.42) HRH1HTR2ACYP2C19LMNACYP19A1
SCHEMBL9899391 0.81 TBXAS1 (0.42) HRH1HTR2ACYP2C19LMNACYP19A1
SCHEMBL1134347 0.81 IDO1 (0.47) IDO1TDO2HRH1HTR2AALDH1A1
SCHEMBL4575392 0.80 HRH1 (0.60) HRH1HTR2AALDH1A1TRPA1SIGMAR1
SCHEMBL9899903 0.80 HTR2A (0.37) HRH1HTR2AALDH1A1OPRK1TRPA1
SCHEMBL9900013 0.79 EPHX2 (0.38) HRH1HTR2AALDH1A1CYP3A4LMNA
SCHEMBL9899816 0.77 SLC6A4 (0.42) HRH1HTR2AALDH1A1TRPA1SIGMAR1
SCHEMBL5410942 0.74 HRH1 (0.58) HRH1HTR2AALDH1A1TRPA1SIGMAR1
SCHEMBL31357687 0.74 SLC18A3 (0.39) IDO1TDO2ALDH1A1CYP3A4ALOX15
SCHEMBL9900221 0.73 HTR2A (0.37) HRH1HTR2AALDH1A1TRPA1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2648714-A2 LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AND USES THEREOF Amira Pharmaceuticals, Inc. (US) 2013-10-16 EP disclosed
WO-2012078593-A2 LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AND USES THEREOF AMIRA PHARMACEUTICALS, INC. (US) 2012-06-14 WO disclosed