SCHEMBL9900221

SCHEMBL9900221

OCCCC(c1ccccc1)c1sccc1Br

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.37
HRH1 P35367 4/20 0.37
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
HSD17B10 Q99714 1/20 0.33
TRPA1 O75762 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
KDM1A O60341 2/20 0.31
GRM2 Q14416 1/20 0.31
GRM3 Q14832 1/20 0.31
LTB4R Q15722 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9899816 0.78 SLC6A4 (0.42) HTR2AHRH1SLC6A4SLC6A3ALDH1A1
SCHEMBL4575392 0.75 HRH1 (0.60) HTR2AHRH1ALDH1A1LMNAHSD17B10
SCHEMBL9899776 0.73 IDO1 (0.42) HTR2AHRH1SLC6A4ALDH1A1LMNA
SCHEMBL9899903 0.72 HTR2A (0.37) HTR2AHRH1SLC6A4ALDH1A1LMNA
SCHEMBL5410942 0.69 HRH1 (0.58) HTR2AHRH1ALDH1A1LMNAHSD17B10
SCHEMBL9915910 0.69 LTB4R (0.53) SLC6A3TRPA1LTB4R
SCHEMBL5412370 0.68 HRH1 (0.56) HTR2AHRH1TRPA1SIGMAR1KDM1A
SCHEMBL1667104 0.68 CTSA (0.48)
SCHEMBL1884939 0.67 LMNA (0.59) HTR2AHRH1ALDH1A1LMNAHSD17B10
SCHEMBL9899391 0.67 TBXAS1 (0.42) HTR2AHRH1SLC6A4SLC6A3LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2648714-A2 LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AND USES THEREOF Amira Pharmaceuticals, Inc. (US) 2013-10-16 EP disclosed
WO-2012078593-A2 LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AND USES THEREOF AMIRA PHARMACEUTICALS, INC. (US) 2012-06-14 WO disclosed