SCHEMBL990135

SCHEMBL990135

CCc1occc(=O)c1OCc1ccccc1

nearest known ligand 0.68

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.68
GAA P10253 1/20 0.68
MAOB P27338 2/20 0.49
POLB P06746 1/20 0.49
MAOA P21397 1/20 0.48
KMT2A Q03164 2/20 0.46
HTT P42858 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
ALDH1A1 P00352 2/20 0.46
HPGD P15428 2/20 0.46
MEN1 O00255 1/20 0.46
KCNA2 P16389 1/20 0.43
KCNA5 P22460 1/20 0.43
KCNA1 Q09470 1/20 0.43
KCNA3 P22001 1/20 0.42
NPC1 O15118 1/20 0.42
NPSR1 Q6W5P4 1/20 0.41
GSTP1 P09211 1/20 0.39
MAPK14 Q16539 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6994111 0.87 LMNA (0.67) LMNAGAAMAOBPOLBMAOA
SCHEMBL18837908 0.85 LMNA (0.64) LMNAGAAMAOBPOLBMAOA
SCHEMBL3565933 0.85 LMNA (0.64) LMNAGAAMAOBPOLBMAOA
SCHEMBL12397417 0.82 LMNA (0.60) LMNAGAAMAOBPOLBMAOA
SCHEMBL81547 0.81 LMNA (1.00) LMNAGAAMAOBPOLBMAOA
SCHEMBL3320803 0.81 GAA (0.59) LMNAGAAMAOBPOLBMAOA
SCHEMBL17228662 0.80 KCNA2 (0.43) LMNAGAAPOLBKMT2AALDH1A1
SCHEMBL16921602 0.79 LMNA (0.68) LMNAGAAMAOBPOLBMAOA
SCHEMBL15452988 0.78 GAA (0.44) LMNAGAAMAOBPOLBMAOA
SCHEMBL1785011 0.78 LMNA (0.56) LMNAGAAMAOBPOLBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 66 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118005558-A Compound, preparation method thereof and application thereof in cigarettes 湖北中烟工业有限责任公司 2024-05-10 CN claimed
CN-116768792-B Cinnamamide-hydroxypyridone derivative, and preparation method and application thereof 浙江工业大学 2024-10-18 CN disclosed
CN-118005558-A Compound, preparation method thereof and application thereof in cigarettes 湖北中烟工业有限责任公司 2024-05-10 CN disclosed
CN-116768792-A Cinnamamide-hydroxypyridone derivative, and preparation method and application thereof 浙江工业大学 2023-09-19 CN disclosed
US-9938240-B2 Fluorinated derivatives of 3-hydroxypyridin-4-ones APOTEX INC. (CA) 2018-04-10 US disclosed
US-9938240-B2 Fluorinated derivatives of 3-hydroxypyridin-4-ones APOTEX INC. (CA) 2018-04-10 US disclosed
US-9938240-B2 Fluorinated derivatives of 3-hydroxypyridin-4-ones APOTEX INC. (CA) 2018-04-10 US disclosed
US-20170247329-A1 \"Fluorinated Derivatives of 3-Hydroxypyridin-4-Ones\ APOTEX TECHNOLOGIES INC. (CA) 2017-08-31 US disclosed
US-20170247329-A1 \"Fluorinated Derivatives of 3-Hydroxypyridin-4-Ones\ APOTEX TECHNOLOGIES INC. (CA) 2017-08-31 US disclosed
US-20170247329-A1 \"Fluorinated Derivatives of 3-Hydroxypyridin-4-Ones\ APOTEX TECHNOLOGIES INC. (CA) 2017-08-31 US disclosed
US-5480894-A 3-hydroxypyridin-4-one derivatives as chelating agents BRITISH TECHNOLOGY GROUP LIMITED (GB) 1996-01-02 US disclosed
EP-0644761-A1 HYDROXYPYRIDIN-4-ONES FOR TREATMENT OF PARASITICAL INFECTIONS BTG INTERNATIONAL LIMITED (GB) 1995-03-29 EP disclosed
EP-0619808-A1 3-HYDROXYPYRIDIN-4-ONE DERIVATIVES AS CHELATING AGENTS BTG INTERNATIONAL LIMITED (GB) 1994-10-19 EP disclosed
WO-1994004498-A1 3-HYDROXYPYRIDIN-4-ONE DERIVATIVES AS CHELATING AGENTS BRITISH TECHNOLOGY GROUP LTD. (GB) 1994-03-03 WO disclosed
WO-1993021919-A1 HYDROXYPYRIDIN-4-ONES FOR TREATMENT OF PARASITICAL INFECTIONS BRITISH TECHNOLOGY GROUP LTD. (GB) 1993-11-11 WO disclosed
US-5256676-A 3-hydroxy-pyridin-4-ones useful for treating parasitic infections BRITISH TECHNOLOGY GROUP LIMITED (GB) 1993-10-26 US disclosed
WO-1992012131-A1 3-HYDROXYPYRIDIN-4-ONE DERIVATIVES AS PHARMACEUTICAL COMPOSITIONS BRITISH TECHNOLOGY GROUP LIMITED (GB) 1992-07-23 WO disclosed
EP-0494754-A1 3-hydroxypyridin-4-one derivatives as pharmaceutical compositions BRITISH TECHNOLOGY GROUP LTD (GB) 1992-07-15 EP disclosed
US-4908371-A Pharmaceuticals CIBA-GEIGY CORPORATION (US) 1990-03-13 US disclosed
EP-0316279-A2 Ester derivatives of azacyclic hydroxycompounds CIBA-GEIGY AG (CH) 1989-05-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170247329-A1 \"Fluorinated Derivatives of 3-Hydroxypyridin-4-Ones\ FH, FECH, FPGS LMNA 2354/4885GAA 547/4885MAOB 513/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.