SCHEMBL9903121

SCHEMBL9903121

O=S(=O)(Oc1cc(-c2cccnc2)n[nH]1)C(F)(F)F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
ALK Q9UM73 1/20 0.50
CYP2D6 P10635 1/20 0.47
CYP2A6 P11509 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2B6 P20813 1/20 0.47
CYP2C19 P33261 1/20 0.47
HPGDS O60760 1/20 0.43
PIM1 P11309 8/20 0.41
PIM3 Q86V86 3/20 0.41
PIM2 Q9P1W9 3/20 0.41
NAMPT P43490 2/20 0.41
METAP2 P50579 1/20 0.40
SIRT3 Q9NTG7 1/20 0.40
CYP19A1 P11511 1/20 0.40
BTK Q06187 1/20 0.38
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2662871 0.78 CA12 (0.51) ALDH1A1CYP1A2BTKHDAC3HDAC4
SCHEMBL9172136 0.75 CA1 (0.51) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2A6
SCHEMBL30300107 0.73 ALDH1A1 (0.63) ALDH1A1CYP1A2CYP3A4ALKCYP2D6
SCHEMBL1436892 0.73 ALDH1A1 (0.63) ALDH1A1CYP1A2CYP3A4ALKCYP2D6
SCHEMBL2645462 0.73 NPC1 (0.44) ALDH1A1CYP1A2CYP3A4BTKSMN1; SMN2
SCHEMBL1459841 0.72 CYP2A6 (0.42) ALDH1A1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL3718580 0.72 PTGS1 (0.46) NAMPTCYP19A1SMN1; SMN2
SCHEMBL29462392 0.72 PTGS1 (0.46) NAMPTCYP19A1SMN1; SMN2
SCHEMBL30207053 0.71 PTGS2 (0.44) CYP19A1
SCHEMBL25871475 0.71 PTGS2 (0.44) CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2648518-A2 PYRAZOLE COMPOUNDS FOR CONTROLLING INVERTEBRATE PESTS BASF SE (DE) 2013-10-16 EP disclosed
US-20130253012-A1 Pyrazole Compounds for Controlling Invertebrate Pests BASF SE (DE) 2013-09-26 US disclosed
WO-2012076704-A2 PYRAZOLE COMPOUNDS FOR CONTROLLING INVERTEBRATE PESTS BASF SE (DE) 2012-06-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130253012-A1 Pyrazole Compounds for Controlling Invertebrate Pests RTN3, RRS1, RTF1 ALDH1A1 3516/4885CYP1A2 234/4885CYP3A4 630/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.