SCHEMBL9172136

SCHEMBL9172136

O=S(=O)(Oc1ccc(-c2cccnc2)cc1)C(F)(F)F

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.51
CA2 P00918 2/20 0.51
CA9 Q16790 2/20 0.51
CA12 O43570 1/20 0.51
MKNK1 Q9BUB5 3/20 0.49
MKNK2 Q9HBH9 3/20 0.49
CYP19A1 P11511 4/20 0.48
CYP3A4 P08684 2/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
CYP2A6 P11509 2/20 0.47
ALDH1A1 P00352 1/20 0.47
CYP1A2 P05177 1/20 0.47
KIF11 P52732 1/20 0.46
CYP11B2 P19099 5/20 0.44
CYP11B1 P15538 3/20 0.44
CYP17A1 P05093 3/20 0.44
CHRM5 P08912 1/20 0.44
NPY5R Q15761 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5532552 0.83 CA2 (0.62) CA1CA2CA9CA12KIF11
SCHEMBL24360466 0.83 CA2 (0.62) CA1CA2CA9CA12KIF11
SCHEMBL835233 0.82 PTGS2 (0.40) CYP19A1CYP3A4CYP2A6CYP1A2CYP11B2
SCHEMBL29462392 0.82 PTGS1 (0.46) CA1CA2CA9CA12CYP19A1
SCHEMBL3718580 0.82 PTGS1 (0.46) CA1CA2CA9CA12CYP19A1
SCHEMBL1713465 0.81 KIF11 (0.55) CA1CA2CA9CA12KIF11
SCHEMBL6801382 0.81 CA2 (0.66) CA1CA2CA9CA12MKNK1
SCHEMBL1805795 0.79 CYP11B1 (0.48) MKNK1MKNK2CYP3A4CYP2D6CYP2C9
SCHEMBL24360467 0.78 CA2 (0.56) CA1CA2CA9CA12KIF11
SCHEMBL1772727 0.78 TBXAS1 (0.43) CYP2D6CYP2A6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0360369-B1 11-Beta-phenyl-14-beta-H-steroids SCHERING AG (DE) 1995-05-03 EP disclosed
EP-0360369-A1 11-Beta-phenyl-14-beta-H-steroids SCHERING AKTIENGESELLSCHAFT (DE) 1990-03-28 EP disclosed