SCHEMBL9904037

SCHEMBL9904037

Cn1c(=O)c2c(nc(-n3cc(-c4ccc(CO)cc4)nn3)n2C)n(C)c1=O

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAOA P21397 7/20 0.47
MAOB P27338 7/20 0.47
GRM2 Q14416 1/20 0.42
RXFP1 Q9HBX9 3/20 0.41
KMT2A Q03164 2/20 0.41
ADORA2A P29274 4/20 0.41
ADORA2B P29275 4/20 0.41
ALDH1A1 P00352 1/20 0.40
PKM P14618 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9904107 0.79 ADORA2B (0.46) KMT2AADORA2AADORA2BALDH1A1
SCHEMBL9904093 0.76 MAOB (0.52) MAOAMAOBRXFP1KMT2AALDH1A1
SCHEMBL9904155 0.70 ADORA2B (0.48) ADORA2AADORA2BALDH1A1
SCHEMBL17091027 0.67 EPHB4 (0.43) KMT2A
SCHEMBL9904038 0.65 MAOB (0.49) MAOAMAOBADORA2AADORA2B
SCHEMBL28061963 0.64 RXFP1 (0.59) MAOAMAOBRXFP1KMT2A
SCHEMBL9904126 0.64 DCTPP1 (0.56) KMT2AADORA2AADORA2BALDH1A1
SCHEMBL9928556 0.62 ADORA2B (0.61) ADORA2AADORA2BALDH1A1PKM
SCHEMBL9904014 0.62 PTGS2 (0.45) KMT2AADORA2AADORA2B
SCHEMBL19449443 0.61 CA2 (0.42) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2465859-A1 8-Triazolylxanthine derivatives, processes for their production and their use as adenosine receptor antagonists Life & Brain GmbH (DE) 2012-06-20 EP disclosed
WO-2012076974-A1 8-TRIAZOLYLXANTHINE DERIVATIVES, PROCESSES FOR THEIR PRODUCTION AND THEIR USE AS ADENOSINE RECEPTOR ANTAGONISTS LIFE & BRAIN GMBH (DE) 2012-06-14 WO disclosed
WO-2012076974-A1 8-TRIAZOLYLXANTHINE DERIVATIVES, PROCESSES FOR THEIR PRODUCTION AND THEIR USE AS ADENOSINE RECEPTOR ANTAGONISTS LIFE & BRAIN GMBH (DE) 2012-06-14 WO disclosed