SCHEMBL9905478

SCHEMBL9905478

O=C(O)NC12CCC(CC1)Cn1c2nc(-c2nc(Cl)c(Cc3ccc(F)cc3)[nH]2)c(OCc2ccccc2)c1=O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.34
ALDH1A1 P00352 2/20 0.33
HPGD P15428 1/20 0.33
CNR2 P34972 1/20 0.32
CHRM4 P08173 1/20 0.32
S1PR5 Q9H228 1/20 0.32
GSK3A P49840 1/20 0.32
GSK3B P49841 1/20 0.32
MAPK14 Q16539 1/20 0.32
USP2 O75604 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
TSHR P16473 1/20 0.31
PRKAA2 P54646 1/20 0.31
MAOA P21397 1/20 0.31
OPRD1 P41143 1/20 0.31
OPRK1 P41145 1/20 0.31
MMP13 P45452 2/20 0.31
HPD P32754 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16130152 0.94 ALDH1A1 (0.34) SMN1; SMN2ALDH1A1HPGDCNR2CHRM4
SCHEMBL9921562 0.87 TLR2 (0.34) ALDH1A1HPGDCNR2MMP13MMP1
SCHEMBL14122561 0.86 MMP13 (0.34) SMN1; SMN2ALDH1A1HPGDCHRM4S1PR5
SCHEMBL9905183 0.83 CNR2 (0.34) SMN1; SMN2ALDH1A1HPGDCNR2USP2
SCHEMBL9905364 0.83 MAPT (0.35) SMN1; SMN2ALDH1A1HPGDCNR2MAOA
SCHEMBL9905325 0.78 SIGMAR1 (0.35) SMN1; SMN2ALDH1A1HPGDCNR2CHRM4
SCHEMBL14214195 0.77 PRSS1 (0.35) SMN1; SMN2ALDH1A1HPGDCNR2MAOA
SCHEMBL14214196 0.77 CNR2 (0.35) SMN1; SMN2ALDH1A1HPGDCNR2CYP1A2
SCHEMBL9905089 0.77 CHRM4 (0.34) SMN1; SMN2ALDH1A1HPGDCNR2CHRM4
SCHEMBL14214198 0.76 ALDH1A1 (0.32) SMN1; SMN2ALDH1A1HPGDUSP2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2649074-A1 HIV INTEGRASE INHIBITORS Bristol-Myers Squibb Company (US) 2013-10-16 EP disclosed
WO-2012078844-A1 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-06-14 WO disclosed