Metformin

Metformin

SCHEMBL991100

CCC(=O)O.CN(C)C(=N)NC(=N)N

nearest known ligand 0.40

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

COXFA4COXFA4L2GPD2MT-ND1MT-ND2MT-ND3MT-ND4MT-ND4LMT-ND5MT-ND6NDUFA1NDUFA10NDUFA11NDUFA12NDUFA13NDUFA2NDUFA3NDUFA5NDUFA6NDUFA7NDUFA8NDUFA9NDUFAB1NDUFAF1NDUFAF2NDUFAF3NDUFAF4NDUFB1NDUFB10NDUFB11NDUFB2NDUFB3NDUFB4NDUFB5NDUFB6NDUFB7NDUFB8NDUFB9NDUFC1NDUFC2NDUFS1NDUFS2NDUFS3NDUFS4NDUFS5NDUFS6NDUFS7NDUFS8NDUFV1NDUFV2NDUFV3

The experimentally established mechanism targets of Metformin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
FFAR3 O14843 1/20 0.40
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Metformin SCHEMBL2231852 0.90 LDHA (0.38) CYP2C19
Metformin SCHEMBL2815239 0.88 LDHA (0.36) CYP2C19
Metformin SCHEMBL7647374 0.88 PHF8 (0.41) FFAR3CYP2C19
Metformin SCHEMBL1558869 0.88 PHF8 (0.41) FFAR3CYP2C19
Metformin SCHEMBL1557197 0.88 GLRA1 (0.40) CYP2C19
Metformin SCHEMBL991940 0.87 FFAR3 (0.46) FFAR3
Metformin SCHEMBL7123890 0.86 PHF8 (0.39)
Metformin SCHEMBL4410446 0.85 CRBN (0.33) FFAR3
Metformin SCHEMBL4364474 0.85 LMNA (0.30)
Metformin SCHEMBL1323029 0.85 CRBN (0.33) FFAR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011008053-A3 PROPIONATE OF N,N-DIMETHYL IMIDOCARBON IMIDIC DIAMIDE, METHOD OF PREPARING SAME, AND PHARMACEUTICAL COMPOSITIONS AND COMBINATIONS CONTAINING SAME 한올바이오파마주식회사 (KR) 2011-04-21 WO disclosed
WO-2011008053-A2 PROPIONATE OF N,N-DIMETHYL IMIDOCARBON IMIDIC DIAMIDE, METHOD OF PREPARING SAME, AND PHARMACEUTICAL COMPOSITIONS AND COMBINATIONS CONTAINING SAME 한올바이오파마주식회사 (KR) 2011-01-20 WO disclosed