SCHEMBL9915426

SCHEMBL9915426

CCCCOc1cc(-c2cc(CN3C(=O)c4ccccc4C3=O)on2)[n+]([O-])cc1OCCCC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
RECQL P46063 2/20 0.48
CYP1A2 P05177 2/20 0.48
CYP2C19 P33261 2/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
HTT P42858 1/20 0.48
CA12 O43570 4/20 0.38
CA9 Q16790 3/20 0.36
CYP19A1 P11511 1/20 0.36
CYP2C9 P11712 1/20 0.36
STAT3 P40763 1/20 0.36
HPGD P15428 4/20 0.35
TSHR P16473 3/20 0.35
RAB9A P51151 2/20 0.35
NPC1 O15118 1/20 0.35
MAPK1 P28482 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PTK2B Q14289 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15275358 0.86 MAPT (0.54) MAPTSMN1; SMN2RECQLCYP1A2CYP2C19
SCHEMBL9915307 0.78 RAB9A (0.43) MAPTSMN1; SMN2HPGDTSHRRAB9A
SCHEMBL9915431 0.78 NOTUM (0.36) CYP1A2CYP2C19CA12CA9CYP19A1
SCHEMBL9915473 0.72 GAA (0.42) TSHR
SCHEMBL9915470 0.71 SMPD1 (0.37) MAPTSMN1; SMN2HTTTSHR
SCHEMBL15279029 0.70 KMT2A (0.41) MAPTSMN1; SMN2HPGDTSHRRAB9A
SCHEMBL9915312 0.68 ALDH1A1 (0.47) MAPTSMN1; SMN2RECQLHPGDTSHR
SCHEMBL14124959 0.66 NOTUM (0.46) SMN1; SMN2STAT3HPGDRAB9ANPC1
SCHEMBL9915495 0.65 SMPD1 (0.41) MAPTRECQLHTTHPGDALDH1A1
SCHEMBL1457566 0.65 MAPT (0.63) MAPTSMN1; SMN2RECQLCYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2646436-B1 MONOBACTAMS PFIZER (US) 2015-05-27 EP disclosed
WO-2012073138-A1 MONOBACTAMS PFIZER INC. (US) 2012-06-07 WO disclosed