SCHEMBL9921565

SCHEMBL9921565

NC12CCC(CC1)Cn1c2nc(-c2ncc(Cc3ccc(F)cc3)[nH]2)c(O)c1=O

nearest known ligand 0.31

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 5/20 0.31
CNR1 P21554 2/20 0.31
CCR2 P41597 1/20 0.31
BRS3 P32247 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14235960 0.85 MMP1 (0.30)
SCHEMBL14214198 0.85 ALDH1A1 (0.32) CCR2BRS3
SCHEMBL9905149 0.83 CCR2 (0.31) CCR2
SCHEMBL9921569 0.83 CYP2C9 (0.35)
SCHEMBL9921570 0.82 CYP2C9 (0.35) CNR2CNR1
SCHEMBL9921578 0.82 CNR2 (0.32) CNR2CNR1
SCHEMBL9921584 0.81 SMN1; SMN2 (0.35) CNR2CNR1
SCHEMBL14214201 0.81 CYP2C9 (0.35) CNR2
SCHEMBL9921583 0.79 RAB9A (0.35) CNR2CNR1
SCHEMBL16130154 0.78 CYP19A1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8846659-B2 HIV integrase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2014-09-30 US disclosed
US-8846659-B2 HIV integrase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2014-09-30 US disclosed
WO-2012078844-A1 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-06-14 WO disclosed