SCHEMBL9923388

SCHEMBL9923388

CN/C=C\C(=N)NC(=O)c1cc(Oc2ccc(C(=O)NCCO)c(F)c2)c2c(c1)OC(C)(C)C2

nearest known ligand 0.49

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GCK P35557 4/20 0.49
EZH2 Q15910 1/20 0.33
FFAR4 Q5NUL3 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9071966 0.89 GCK (0.53) GCKEZH2
SCHEMBL2669358 0.88 GCK (0.46) GCK
SCHEMBL2669236 0.87 GCK (0.49) GCKEZH2
SCHEMBL2669283 0.85 GCK (0.66) GCKEZH2
SCHEMBL2643748 0.85 GCK (0.54) GCKEZH2FFAR4
SCHEMBL2669286 0.84 GCK (0.55) GCK
SCHEMBL2669365 0.83 GCK (0.46) GCKFFAR4
SCHEMBL2669296 0.82 GCK (0.41) GCK
SCHEMBL2669367 0.82 GCK (0.55) GCKEZH2
SCHEMBL9071945 0.82 GCK (0.55) GCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2463283-A1 Fused phenyl Amido heterocyclic compounds for the prevention and treatment of glucokinase-mediated diseases Pfizer Products Inc. (US) 2012-06-13 EP disclosed