SCHEMBL9923403

SCHEMBL9923403

C/C=C/N=C(\CC)NC(=O)c1cc(Oc2ccc(C(=O)N(C)C)c(F)c2)c2c(c1)OC(C)(C)C2

nearest known ligand 0.49

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GCK P35557 4/20 0.49
EZH2 Q15910 1/20 0.30
SCN9A Q15858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2669366 0.82 GCK (0.50) GCKEZH2SCN9A
SCHEMBL2669236 0.81 GCK (0.49) GCKEZH2
SCHEMBL643703 0.81 GCK (0.53) GCKEZH2SCN9A
SCHEMBL644377 0.80 GCK (0.52) GCKEZH2
SCHEMBL643421 0.78 GCK (0.56) GCK
SCHEMBL12101417 0.77 GCK (0.47) GCKEZH2
SCHEMBL642567 0.77 GCK (0.59) GCK
SCHEMBL643673 0.77 GCK (0.59) GCK
SCHEMBL643599 0.76 GCK (0.65) GCK
SCHEMBL643823 0.76 GCK (0.78) GCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2463283-A1 Fused phenyl Amido heterocyclic compounds for the prevention and treatment of glucokinase-mediated diseases Pfizer Products Inc. (US) 2012-06-13 EP disclosed