SCHEMBL9933014

SCHEMBL9933014

Nc1cc(Cl)c(O)c(Br)c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.68
CYP3A4 P08684 6/20 0.46
ALDH1A1 P00352 2/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
CA1 P00915 3/20 0.43
CA2 P00918 3/20 0.43
ERN1 O75460 1/20 0.41
TSHR P16473 5/20 0.40
HSD17B10 Q99714 4/20 0.40
TTR P02766 3/20 0.40
TDP1 Q9NUW8 1/20 0.40
RECQL P46063 1/20 0.40
HPGD P15428 2/20 0.37
CA4 P22748 1/20 0.37
CA6 P23280 1/20 0.37
MAPK1 P28482 1/20 0.37
TP53 P04637 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL95180 0.82 CYP3A4 (0.58) THRBCYP3A4ALDH1A1GAAMAPT
SCHEMBL93999 0.82 THRB (1.00) THRBCYP3A4ALDH1A1GAAMAPT
Hydrochloric Acid SCHEMBL4929431 0.79 CYP3A4 (0.55) THRBCYP3A4ALDH1A1GAAMAPT
Hydrochloric Acid SCHEMBL7755405 0.79 THRB (0.94) THRBCYP3A4ALDH1A1GAAMAPT
Hydrochloric Acid SCHEMBL10336483 0.79 THRB (0.94) THRBCYP3A4ALDH1A1GAAMAPT
SCHEMBL9453347 0.79 THRB (0.94) THRBCYP3A4ALDH1A1GAAMAPT
SCHEMBL5271617 0.79 THRB (0.94) THRBCYP3A4ALDH1A1GAAMAPT
SCHEMBL2417306 0.77 TSHR (0.68) THRBCYP3A4ALDH1A1MAPTCA1
Hydrochloric Acid SCHEMBL10336482 0.75 THRB (0.84) THRBCYP3A4ALDH1A1GAAMAPT
SCHEMBL21695780 0.75 GAA (0.50) THRBCYP3A4ALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122036699-A THR-beta modulators and methods of use thereof 阿利戈斯治疗公司 2026-05-15 CN disclosed
US-20250304561-A1 MODULATORS OF THR-BETA AND METHODS OF USE THEREOF ALIGOS THERAPEUTICS, INC. (US) 2025-10-02 US disclosed
EP-4523692-A2 MODULATORS OF THR-SS AND METHODS OF USE THEREOF Aligos Therapeutics, Inc. (US) 2025-03-19 EP disclosed
EP-3965884-B1 MODULATORS OF THR-BETA WITH A DIOXO-1,2,4-TRIAZYL HEAD GROUP ALIGOS THERAPEUTICS INC (US) 2025-01-15 EP disclosed
US-12180192-B2 Modulators of THR-β and methods of use thereof ALIGOS THERAPEUTICS, INC. (US) 2024-12-31 US disclosed
US-11926618-B2 Halogen-substituted phenylate compound and applications thereof HINOVA PHARMACEUTICALS INC. (CN) 2024-03-12 US disclosed
US-20220332707-A1 HALOGEN-SUBSTITUTED PHENYLATE COMPOUND AND APPLICATIONS THEREOF HINOVA PHARMACEUTICALS INC. (CN) 2022-10-20 US disclosed
EP-4019510-A1 HALOGEN-SUBSTITUTED PHENYLATE COMPOUND AND APPLICATIONS THEREOF Hinova Pharmaceuticals Inc. (CN) 2022-06-29 EP disclosed
EP-4019510-A1 HALOGEN-SUBSTITUTED PHENYLATE COMPOUND AND APPLICATIONS THEREOF Hinova Pharmaceuticals Inc. (CN) 2022-06-29 EP disclosed
CN-112409340-B Halogen substituted phenyl ether compound and application thereof 海创药业股份有限公司 2022-03-18 CN disclosed
US-11091467-B2 Modulators of THR-β and methods of use thereof ALIGOS THERAPEUTICS, INC. (US) 2021-08-17 US disclosed
CN-112409340-A Halogen substituted phenyl ether compound and application thereof 海创药业股份有限公司 2021-02-26 CN disclosed
WO-2021032161-A1 HALOGEN-SUBSTITUTED PHENYLATE COMPOUND AND APPLICATIONS THEREOF 成都海创药业有限公司 2021-02-25 WO disclosed
WO-2021032161-A1 HALOGEN-SUBSTITUTED PHENYLATE COMPOUND AND APPLICATIONS THEREOF 成都海创药业有限公司 2021-02-25 WO disclosed
WO-2020239076-A1 PYRIDAZINONE DERIVATIVES AS THYROXINE RECEPTOR-Β AGONISTS AND APPLICATION THEREOF 南京明德新药研发有限公司 2020-12-03 WO disclosed
WO-2020227549-A1 MODULATORS OF THR-β AND METHODS OF USE THEREOF ALIGOS THERAPEUTICS, INC. (US) 2020-11-12 WO disclosed
US-20200354345-A1 MODULATORS OF THR-BETA AND METHODS OF USE THEREOF ALIGOS THERAPEUTICS, INC. (US) 2020-11-12 US disclosed
US-20120157482-A1 COMPOUNDS AND METHODS GLAXOSMITHKLINE LLC 2012-06-21 US disclosed
US-4675290-A CHROMATOGRAPHY OF THE ANILINE DYE PRODUCED BY COUPLING REACTI ON OF THE AMINE FORMED FROM THE AMIDE SUBSTRATE TOYO JOZO KABUSHIKI KAISHA (JP) 1987-06-23 US disclosed
US-4588836-A LEUCYL- OR GLUTAMYL-3,5-DIHALO-4-HYDROXYANILIDES TOYO JOZO KABUSHIKI KAISHA (JP) 1986-05-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11926618-B2 Halogen-substituted phenylate compound and applications thereof THRB, FFAR3, THRA THRB 1/4885CYP3A4 168/4885ALDH1A1 2721/4885
US-20250304561-A1 MODULATORS OF THR-BETA AND METHODS OF USE THEREOF THRB, THRA, TRHR THRB 1/4885CYP3A4 3296/4885ALDH1A1 3330/4885
US-20200354345-A1 MODULATORS OF THR-BETA AND METHODS OF USE THEREOF THRB, THRA, TRHR THRB 1/4885CYP3A4 3790/4885ALDH1A1 3081/4885
US-20220332707-A1 HALOGEN-SUBSTITUTED PHENYLATE COMPOUND AND APPLICATIONS THEREOF THRB, FFAR3, THRA THRB 1/4885CYP3A4 168/4885ALDH1A1 2721/4885
US-12180192-B2 Modulators of THR-β and methods of use thereof THRB, THRA, TRHR THRB 1/4885CYP3A4 3759/4885ALDH1A1 3049/4885
US-20120157482-A1 COMPOUNDS AND METHODS NQO1, CYP1B1, CYP1A1 THRB 2458/4885CYP3A4 23/4885ALDH1A1 52/4885
US-11091467-B2 Modulators of THR-β and methods of use thereof THRB, THRA, TRHR THRB 1/4885CYP3A4 3759/4885ALDH1A1 3049/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.