SCHEMBL9938769

SCHEMBL9938769

COc1ccc(CNC(=O)NC[C@H]2OC(O)[C@H](NC(=O)c3cccc(-c4ccccc4)c3)[C@@H](O)[C@@H]2O)cc1

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HK1 P19367 12/20 0.60
HK2 P52789 12/20 0.60
GCK P35557 1/20 0.55
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
HPGD P15428 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
SENP1 Q9P0U3 2/20 0.44
MAPK1 P28482 1/20 0.43
EPHX2 P34913 1/20 0.43
NR1H4 Q96RI1 1/20 0.43
ERN1 O75460 1/20 0.43
CD22 P20273 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9938774 1.00 HK1 (0.60) HK1HK2GCKNPC1RAB9A
SCHEMBL9937930 0.87 HK1 (0.46) HK1HK2GCKNPC1RAB9A
SCHEMBL9971331 0.83 HK1 (0.73) HK1HK2GCK
SCHEMBL9937688 0.78 HK1 (0.69) HK1HK2GCKEPHX2NR1H4
SCHEMBL9937695 0.78 HK1 (0.69) HK1HK2GCKEPHX2NR1H4
SCHEMBL9971381 0.76 ALDH1A1 (0.41) HK1HK2NPC1RAB9AKDM4E
SCHEMBL1926645 0.76 NPC1 (0.78) NPC1RAB9AKDM4EALDH1A1HPGD
SCHEMBL9937446 0.76 HK1 (1.00) HK1HK2GCK
SCHEMBL9937441 0.76 HK1 (1.00) HK1HK2GCK
SCHEMBL9938423 0.72 HK2 (0.80) HK1HK2GCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012083145-A1 GLUCOSAMINE DERIVATIVES GLAXO WELLCOME MANUFACTURING PTE LTD (SG) 2012-06-21 WO disclosed