SCHEMBL9952084

SCHEMBL9952084

COc1c(CCCOC(N)=O)cc(Cl)c(C)c1Br

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.38
IMPDH2 P12268 2/20 0.37
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 2/20 0.37
GAA P10253 1/20 0.37
SLC2A1 P11166 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
TSHR P16473 2/20 0.31
APOBEC3A P31941 1/20 0.31
HTT P42858 1/20 0.31
APOBEC3G Q9HC16 1/20 0.31
HSP90AA1 P07900 1/20 0.31
NPSR1 Q6W5P4 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
NCOA1 Q15788 1/20 0.30
NCOA3 Q9Y6Q9 1/20 0.30
CA1 P00915 2/20 0.30
CA2 P00918 2/20 0.30
CA12 O43570 1/20 0.30
CA9 Q16790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9952278 0.92 ALDH1A1 (0.38) LMNAIMPDH2ALDH1A1KDM4EGAA
SCHEMBL9953183 0.80 TAAR1 (0.37) IMPDH2ALDH1A1KDM4EGAASLC2A1
SCHEMBL9952087 0.77 IMPDH2 (0.38) IMPDH2ALDH1A1KDM4EGAASLC2A1
SCHEMBL9952029 0.77 TAAR1 (0.46) IMPDH2
Hydrochloric Acid SCHEMBL9952054 0.76 TAAR1 (0.45) IMPDH2
SCHEMBL9952473 0.75 IMPDH2 (0.41) LMNAIMPDH2ALDH1A1KDM4EGAA
SCHEMBL14742274 0.75 IMPDH2 (0.36) IMPDH2SLC2A1CA1CA2
SCHEMBL28712872 0.75 ALDH1A1 (0.44) LMNAIMPDH2ALDH1A1KDM4EGAA
SCHEMBL9953040 0.74 IMPDH2 (0.45) LMNAIMPDH2ALDH1A1KDM4EGAA
SCHEMBL9953206 0.73 IMPDH2 (0.34) IMPDH2ALDH1A1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655374-A1 N-(1-(SUBSTITUTED-PHENYL)ETHYL)-9H-PURIN-6-AMINES AS PI3K INHIBITORS Incyte Corporation (US) 2013-10-30 EP disclosed
WO-2012087881-A1 N-(1-(SUBSTITUTED-PHENYL)ETHYL)-9H-PURIN-6-AMINES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2012-06-28 WO disclosed