SCHEMBL9952473

SCHEMBL9952473

COc1c(CCNC(=O)O)cc(Cl)c(C)c1Br

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 1/20 0.41
SLC2A1 P11166 1/20 0.40
SHMT2 P34897 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KMT2A Q03164 2/20 0.38
POLB P06746 1/20 0.38
MTNR1A P48039 4/20 0.37
MTNR1B P49286 4/20 0.37
MEN1 O00255 1/20 0.37
LMNA P02545 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
NFKB1 P19838 1/20 0.37
MAPK1 P28482 1/20 0.37
SLC6A4 P31645 1/20 0.37
CYP2C19 P33261 1/20 0.37
THPO P40225 1/20 0.37
HTR2B P41595 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9952754 0.81 IMPDH2 (0.42) IMPDH2SLC2A1SHMT2KMT2APOLB
SCHEMBL9952087 0.80 IMPDH2 (0.38) IMPDH2SLC2A1KMT2ACYP1A2CYP3A4
SCHEMBL14742274 0.78 IMPDH2 (0.36) IMPDH2SLC2A1
SCHEMBL9952992 0.78 IMPDH2 (0.37) IMPDH2SLC2A1SHMT2KMT2AMTNR1A
SCHEMBL9952278 0.77 ALDH1A1 (0.38) IMPDH2SLC2A1SMN1; SMN2KMT2AMEN1
SCHEMBL9953040 0.77 IMPDH2 (0.45) IMPDH2POLBMTNR1AMTNR1BLMNA
SCHEMBL9952029 0.77 TAAR1 (0.46) IMPDH2CYP1A2HTR2B
SCHEMBL9952243 0.76 IMPDH2 (0.36) IMPDH2SLC2A1SHMT2KMT2AMTNR1A
Hydrochloric Acid SCHEMBL9952054 0.76 TAAR1 (0.45) IMPDH2CYP1A2HTR2B
SCHEMBL9952084 0.75 LMNA (0.38) IMPDH2SLC2A1SMN1; SMN2LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655374-A1 N-(1-(SUBSTITUTED-PHENYL)ETHYL)-9H-PURIN-6-AMINES AS PI3K INHIBITORS Incyte Corporation (US) 2013-10-30 EP disclosed
WO-2012087881-A1 N-(1-(SUBSTITUTED-PHENYL)ETHYL)-9H-PURIN-6-AMINES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2012-06-28 WO disclosed