SCHEMBL9953300

SCHEMBL9953300

Nc1nc2ccc(Br)cc2c(=O)n1CC1CC1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 3/20 0.46
PDE4A P27815 3/20 0.46
PDE4B Q07343 3/20 0.46
PDE4C Q08493 3/20 0.46
PDE4D Q08499 3/20 0.46
CACNA2D1 P54289 5/20 0.44
CTSD P07339 6/20 0.44
MAPK8 P45983 2/20 0.44
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
ATM Q13315 1/20 0.41
CYP3A4 P08684 1/20 0.41
DPP4 P27487 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31241110 1.00 PDE5A (0.46) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL31241042 0.85 MAPK8 (0.47) CACNA2D1MAPK8MEN1KMT2AATM
SCHEMBL31241091 0.81 CACNA2D1 (0.47) CACNA2D1MEN1KMT2AATMALDH1A1
SCHEMBL20641274 0.81 AURKA (0.47) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL10289136 0.81 CACNA2D1 (0.51) CACNA2D1MEN1KMT2AATMHTT
SCHEMBL10289135 0.80 CTSD (0.48) CACNA2D1CTSDALDH1A1HTT
SCHEMBL9955787 0.78 CTSD (0.47) CACNA2D1CTSDALDH1A1HTT
SCHEMBL9029528 0.77 TP53 (0.47) CACNA2D1MAPK8ATMALDH1A1
SCHEMBL9952969 0.77 DPP4 (0.51) CACNA2D1MEN1KMT2AATMDPP4
SCHEMBL10288755 0.77 POLR1A (0.41) CACNA2D1CTSDALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed