SCHEMBL9955787

SCHEMBL9955787

Nc1nc2ccc(Br)cc2c(=O)n1CC1CNCCO1

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSD P07339 8/20 0.47
ALDH1A1 P00352 1/20 0.42
HTT P42858 1/20 0.42
CACNA2D1 P54289 6/20 0.41
OPRM1 P35372 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10289135 0.83 CTSD (0.48) CTSDALDH1A1HTTCACNA2D1
SCHEMBL31241110 0.78 PDE5A (0.46) CTSDALDH1A1HTTCACNA2D1
SCHEMBL9953300 0.78 PDE5A (0.46) CTSDALDH1A1HTTCACNA2D1
SCHEMBL28228572 0.74 LMNA (0.42) ALDH1A1HTT
SCHEMBL10288755 0.73 POLR1A (0.41) CTSDALDH1A1HTTCACNA2D1OPRM1
SCHEMBL31241091 0.73 CACNA2D1 (0.47) ALDH1A1CACNA2D1OPRM1
SCHEMBL10289136 0.72 CACNA2D1 (0.51) HTTCACNA2D1OPRM1
SCHEMBL9953779 0.72 ALOX15 (0.55) ALDH1A1HTTCACNA2D1
SCHEMBL9960599 0.70 MAPK1 (0.49) ALDH1A1HTT
SCHEMBL9952969 0.69 DPP4 (0.51) ALDH1A1CACNA2D1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed