SCHEMBL9953968

SCHEMBL9953968

Cc1ccc(-c2ccccc2)c(C=O)n1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
S100A4 P26447 1/20 0.39
TGFBR1 P36897 1/20 0.37
HTR2B P41595 1/20 0.37
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
KDM4C Q9H3R0 1/20 0.36
PSMB5 P28074 1/20 0.36
DHODH Q02127 3/20 0.35
CYP1A2 P05177 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
AKT1 P31749 1/20 0.35
AKT2 P31751 1/20 0.35
ESR2 Q92731 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13309126 0.82 ADORA2A (0.39) S100A4TGFBR1ADORA2AADORA1DHODH
SCHEMBL16279826 0.82 CYP2A6 (0.53) CYP1A2
SCHEMBL28132406 0.80 ALDH1A1 (0.44) HTR2BPSMB5CYP1A2L3MBTL1GAA
SCHEMBL29956107 0.78 ASIC3 (0.41) ADORA2AADORA1
SCHEMBL9955665 0.76 S100A4 (0.38) S100A4HTR2B
SCHEMBL29912137 0.76 S100A4 (0.38) S100A4HTR2B
SCHEMBL9955492 0.76 NPC1 (0.46) TGFBR1CYP1A2L3MBTL1GAA
SCHEMBL10262765 0.74 PSMB5 (0.47) TGFBR1ADORA2AADORA1PSMB5CYP1A2
SCHEMBL5360517 0.72 SYK (0.45) S100A4TGFBR1ADORA1PSMB5DHODH
SCHEMBL27852466 0.72 SQOR (0.54) ADORA1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085857-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-3-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed