SCHEMBL9954063

SCHEMBL9954063

Nc1ccc(Br)cc1C(=O)Nc1ccncc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 4/20 0.54
TYK2 P29597 4/20 0.54
HTT P42858 3/20 0.52
PRKCI P41743 3/20 0.52
ALDH1A1 P00352 2/20 0.52
ROCK2 O75116 1/20 0.52
GAA P10253 1/20 0.52
ALOX12 P18054 1/20 0.52
ROCK1 Q13464 1/20 0.52
NPSR1 Q6W5P4 2/20 0.52
CYP3A4 P08684 2/20 0.52
CYP1A2 P05177 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
KDM4E B2RXH2 2/20 0.51
GLA P06280 1/20 0.51
LMNA P02545 1/20 0.49
PTPN7 P35236 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5925259 0.87 MAPT (0.59) HTTALDH1A1GAACYP1A2CYP2C9
SCHEMBL10289025 0.84 POLB (0.61) HTTALDH1A1KDM4EGLASORT1
SCHEMBL6034144 0.83 SORT1 (0.72) ALDH1A1KDM4ESORT1KMT2ANPC1
SCHEMBL5925289 0.82 KDM4E (0.51) HTTALDH1A1GAACYP1A2CYP2C9
SCHEMBL7516613 0.82 HDAC1 (0.64) HTTALDH1A1GAACYP1A2CYP2C9
SCHEMBL26758014 0.79 SMN1; SMN2 (0.76) JAK2TYK2HTTALDH1A1GAA
SCHEMBL14059394 0.79 PRKCI (0.66) HTTPRKCIALDH1A1ROCK2GAA
SCHEMBL460200 0.78 PRKCI (0.67) JAK2TYK2HTTPRKCIALDH1A1
SCHEMBL30339468 0.78 PRKCI (0.67) JAK2TYK2HTTPRKCIALDH1A1
SCHEMBL14917439 0.78 ROCK2 (0.66) JAK2TYK2HTTPRKCIALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed