SCHEMBL14917439

SCHEMBL14917439

Nc1ccncc1C(=O)Nc1ccncc1

nearest known ligand 0.66

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.66
ROCK1 Q13464 2/20 0.66
PRKCI P41743 3/20 0.58
TYK2 P29597 5/20 0.55
JAK2 O60674 5/20 0.55
KDM4E B2RXH2 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
HTT P42858 2/20 0.53
JAK1 P23458 3/20 0.51
GAA P10253 2/20 0.51
NCOA1 Q15788 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
NCOA3 Q9Y6Q9 1/20 0.51
MDM2 Q00987 1/20 0.50
POLB P06746 1/20 0.50
MAPT P10636 1/20 0.50
ALDH1A1 P00352 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14917461 0.90 PRKCI (0.56) ROCK2ROCK1PRKCITYK2JAK2
SCHEMBL14917435 0.85 ALDH1A1 (0.61) PRKCIKDM4EHTTALDH1A1
SCHEMBL30339468 0.83 PRKCI (0.67) PRKCITYK2JAK2HTTJAK1
SCHEMBL460200 0.83 PRKCI (0.67) PRKCITYK2JAK2HTTJAK1
SCHEMBL15140751 0.79 ROCK2 (1.00) ROCK2ROCK1TYK2JAK2KDM4E
Ammonia Solution, Strong SCHEMBL27706531 0.79 GAA (0.50) ROCK2ROCK1KDM4EL3MBTL1GAA
SCHEMBL1232259 0.79 GAA (0.50) ROCK2ROCK1KDM4EL3MBTL1GAA
SCHEMBL9954063 0.78 JAK2 (0.54) ROCK2ROCK1PRKCITYK2JAK2
SCHEMBL16713265 0.78 CHRNB2 (0.55) ROCK2ROCK1PRKCIKDM4EL3MBTL1
SCHEMBL14917446 0.76 NPC1 (0.67) KDM4ESMN1; SMN2MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130116430-A1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF FUJIFILM CORPORATION (JP) 2013-05-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130116430-A1 NOVEL NICOTINAMIDE DERIVATIVE OR SALT THEREOF SYK, CD38, BTK ROCK2 1485/4885ROCK1 849/4885PRKCI 748/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.