SCHEMBL9954750

SCHEMBL9954750

Nc1cc(Br)cc2oc(=O)[nH]c12

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.37
KMO O15229 1/20 0.35
MCL1 Q07820 1/20 0.35
GPR35 Q9HC97 1/20 0.34
NOS1 P29475 4/20 0.33
NOS3 P29474 3/20 0.33
NOS2 P35228 3/20 0.33
OGT O15294 1/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
ADRA2A P08913 1/20 0.33
TSHR P16473 1/20 0.33
THPO P40225 1/20 0.33
BLM P54132 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
IDO1 P14902 1/20 0.30
TDO2 P48775 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10780521 0.81 GRM5 (0.38) GRM5KMOMCL1GPR35NOS1
SCHEMBL11040536 0.78 NOS1 (0.49) GRM5KMOMCL1NOS1NOS3
SCHEMBL18107837 0.78 GRM5 (0.37) GRM5KMOMCL1NOS1NOS3
SCHEMBL15319641 0.78 KMO (0.47) GRM5KMOMCL1NOS1NOS3
SCHEMBL1285298 0.78 NOS1 (0.41) GRM5KMOMCL1NOS1NOS3
SCHEMBL11040319 0.76 KMO (0.34) KMOMCL1NOS1NOS3NOS2
SCHEMBL18188179 0.74 GAA (0.41) GRM5KMOMCL1NOS1NOS3
SCHEMBL11282616 0.74 MCL1 (0.33) KMOMCL1NOS1NOS3NOS2
SCHEMBL9954720 0.73 GPR35 (0.40) GRM5GPR35LMNACYP1A2TSHR
SCHEMBL11040962 0.70 NOS1 (0.32) KMOMCL1NOS1NOS3NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed