SCHEMBL9954766

SCHEMBL9954766

COc1ncc(B2OC(C)(C)C(C)(C)O2)cc1S(=O)(=O)NC1CCC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALPL P05186 1/20 0.56
PIK3C3 Q8NEB9 2/20 0.48
BRD4 O60885 3/20 0.41
BRD3 Q15059 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
HTT P42858 2/20 0.40
ALDH1A1 P00352 1/20 0.40
MCOLN3 Q8TDD5 1/20 0.40
TP53 P04637 1/20 0.39
CASP1 P29466 1/20 0.39
BRD2 P25440 1/20 0.38
PIK3C2G O75747 2/20 0.38
PIK3CG P48736 2/20 0.38
PIK3CA P42336 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.36
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9953817 0.98 ALPL (0.56) ALPLPIK3C3BRD4BRD3SMN1; SMN2
SCHEMBL9954287 0.97 ALPL (0.55) ALPLPIK3C3BRD4BRD3SMN1; SMN2
SCHEMBL9953730 0.96 ALPL (0.57) ALPLPIK3C3BRD4BRD3SMN1; SMN2
SCHEMBL9953577 0.92 ALPL (0.54) ALPLPIK3C3BRD4BRD3SMN1; SMN2
SCHEMBL21760716 0.91 ALPL (0.53) ALPLPIK3C3BRD4BRD3BRD2
SCHEMBL19303685 0.91 ALPL (0.53) ALPLPIK3C3BRD4BRD3BRD2
SCHEMBL23758152 0.86 ALPL (0.49) ALPLPIK3C3BRD4BRD3SMN1; SMN2
SCHEMBL9953472 0.83 ALPL (0.62) ALPLPIK3C3PIK3CGPIK3CAL3MBTL1
SCHEMBL9952979 0.82 ALPL (0.53) ALPLSMN1; SMN2HTTALDH1A1PIK3CA
SCHEMBL9953660 0.82 ALPL (0.59) ALPLPIK3C3SMN1; SMN2ALDH1A1PIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012174312-A2 BENZIMIDAZOLE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-12-20 WO disclosed
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed