SCHEMBL9954835

SCHEMBL9954835

O=C(Nc1cccnc1)Nc1ccc(Br)cn1

nearest known ligand 0.68

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.68
RAB9A P51151 9/20 0.62
NPC1 O15118 7/20 0.62
MEN1 O00255 3/20 0.59
KMT2A Q03164 3/20 0.59
HTT P42858 2/20 0.59
KDM4E B2RXH2 1/20 0.59
MAPK1 P28482 1/20 0.59
CYP11B1 P15538 1/20 0.57
CYP11B2 P19099 1/20 0.57
POLB P06746 2/20 0.56
MAPT P10636 4/20 0.55
FPR2 P25090 2/20 0.55
ALDH1A1 P00352 2/20 0.54
LMNA P02545 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
TAAR1 Q96RJ0 1/20 0.52
P2RX4 Q99571 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9954640 0.85 RAB9A (0.73) TSHRRAB9ANPC1MEN1KMT2A
SCHEMBL9954182 0.84 RAB9A (0.71) TSHRRAB9ANPC1MEN1KMT2A
SCHEMBL22926672 0.83 FPR2 (0.74) RAB9ANPC1MEN1KMT2AHTT
SCHEMBL29517932 0.83 FPR2 (0.74) RAB9ANPC1MEN1KMT2AHTT
SCHEMBL9637653 0.81 MEN1 (0.77) TSHRRAB9ANPC1MEN1KMT2A
SCHEMBL30051982 0.81 MEN1 (0.77) TSHRRAB9ANPC1MEN1KMT2A
Bromide SCHEMBL29417998 0.79 MEN1 (0.74) TSHRRAB9ANPC1MEN1KMT2A
Hydrochloric Acid SCHEMBL29388210 0.79 MEN1 (0.74) TSHRRAB9ANPC1MEN1KMT2A
SCHEMBL20172471 0.79 NPC1 (0.47) RAB9ANPC1MEN1KMT2AHTT
SCHEMBL31241036 0.78 RAB9A (0.71) RAB9ANPC1MEN1KMT2AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed