SCHEMBL99550

SCHEMBL99550

CN1CCC(N(C(=O)O)c2cc(CCC(=O)Nc3ccc(CO[Si](C)(C)C(C)(C)C)cc3)ccc2-c2ccccc2)CC1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 2/20 0.40
EPHX2 P34913 2/20 0.39
CDK8 P49336 1/20 0.36
ABCB1 P08183 1/20 0.36
MAPT P10636 2/20 0.35
NPC1 O15118 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ROCK2 O75116 1/20 0.35
KDM4E B2RXH2 1/20 0.35
PKM P14618 1/20 0.35
SLC2A1 P11166 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
ALDH1A1 P00352 1/20 0.35
RAB9A P51151 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL661774 0.94 MCHR1 (0.41) MCHR1CDK8MAPTKDM4EPKM
SCHEMBL661325 0.90 PDCD1 (0.36) MCHR1CDK8MAPTROCK2KDM4E
SCHEMBL661903 0.88 S1PR1 (0.34) MCHR1CDK8NPC1PKMRAB9A
SCHEMBL175794 0.87 CDK8 (0.42) MCHR1CDK8ROCK2
SCHEMBL660644 0.86 NPC1 (0.38) MAPTNPC1SMN1; SMN2ROCK2ALDH1A1
SCHEMBL101815 0.86 ALPL (0.37) ALDH1A1
SCHEMBL169855 0.83 CHRM3 (0.51)
SCHEMBL99012 0.81 CHRM3 (0.51)
SCHEMBL132389 0.80 CHEK1 (0.37) SMN1; SMN2
SCHEMBL134109 0.80 ALPL (0.36) SMN1; SMN2HDAC1HDAC2ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426121-A1 QUATERNARY AMMONIUM SALT COMPOUND Teijin Pharma Limited (JP) 2012-03-07 EP claimed