SCHEMBL661774

SCHEMBL661774

CN1CCC(N(C(=O)O)c2cc(CCC(=O)Nc3ccc4cc(CO[Si](C)(C)C(C)(C)C)ccc4c3)ccc2-c2ccccc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 12/20 0.41
CDK8 P49336 1/20 0.37
HCAR2 Q8TDS4 5/20 0.37
KDM4E B2RXH2 1/20 0.36
PKM P14618 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
HTT P42858 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL99550 0.94 MCHR1 (0.40) MCHR1CDK8KDM4EPKMALDH1A1
SCHEMBL661325 0.86 PDCD1 (0.36) MCHR1CDK8KDM4EPKMALDH1A1
SCHEMBL175794 0.85 CDK8 (0.42) MCHR1CDK8
SCHEMBL661903 0.85 S1PR1 (0.34) MCHR1CDK8PKM
SCHEMBL101815 0.84 ALPL (0.37) HCAR2MEN1ALDH1A1KMT2A
SCHEMBL99851 0.84 CHRM3 (0.48)
SCHEMBL660644 0.82 NPC1 (0.38) MEN1ALDH1A1MAPTHTTKMT2A
SCHEMBL663422 0.80 CHRM3 (0.47)
SCHEMBL99078 0.80 HCAR2 (0.42) MCHR1HCAR2MEN1ALDH1A1LMNA
SCHEMBL134109 0.77 ALPL (0.36) MEN1ALDH1A1LMNAHPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120046467-A1 QUATERNARY AMMONIUM SALT COMPOUNDS TEIJIN PHARMA LIMITED (JP) 2012-02-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120046467-A1 QUATERNARY AMMONIUM SALT COMPOUNDS ADRB2, AGTR2, ADRB3 MCHR1 223/4885CDK8 4493/4885HCAR2 42/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.