SCHEMBL9955232

SCHEMBL9955232

COC(OC)c1nc(Cl)oc1-c1cccc(F)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.38
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38
PDGFRB P09619 1/20 0.36
PDGFRA P16234 1/20 0.36
ALDH1A1 P00352 1/20 0.35
CYP1A1 P04798 2/20 0.35
CYP1A2 P05177 2/20 0.35
CYP1B1 Q16678 2/20 0.35
MGAM O43451 1/20 0.35
GAA P10253 1/20 0.35
SI P14410 1/20 0.35
MGAM2 Q2M2H8 1/20 0.35
MAOB P27338 1/20 0.34
XPO1 O14980 1/20 0.34
NOTUM Q6P988 2/20 0.34
NR4A1 P22736 1/20 0.34
NR4A2 P43354 1/20 0.34
NR4A3 Q92570 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9956151 0.83 KDM4E (0.42) KDM4EMEN1MAPTKMT2AALDH1A1
SCHEMBL9955368 0.77 KDM4E (0.41) KDM4EMEN1MAPTKMT2AALDH1A1
SCHEMBL11750022 0.75 KDM4E (0.41) KDM4EMEN1MAPTKMT2AALDH1A1
SCHEMBL9956192 0.75 MAPK14 (0.42) KDM4EMAPTPDGFRBPDGFRACYP1A1
SCHEMBL11750444 0.73 RXRA (0.45) KDM4EMEN1MAPTKMT2ACYP1A2
SCHEMBL9955896 0.70 NOTUM (0.39) KDM4EMEN1MAPTKMT2AALDH1A1
SCHEMBL9955196 0.70 L3MBTL1 (0.45) KDM4EMEN1MAPTKMT2AALDH1A1
SCHEMBL11755076 0.70 ADORA2A (0.46) KDM4EMEN1MAPTKMT2AALDH1A1
SCHEMBL10263245 0.69 TRPM8 (0.42) MGAMGAASIMGAM2MAOB
SCHEMBL9954109 0.68 ADORA2A (0.45) KDM4EMEN1MAPTKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085852-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-8-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed
WO-2012085852-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-8-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed
WO-2012085857-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-3-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed
WO-2012085857-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-3-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed