SCHEMBL9956809

SCHEMBL9956809

C=CCc1[nH]c(C)c(C(=O)Cl)c1C

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.43
NPSR1 Q6W5P4 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
HPGD P15428 2/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
ALOX15 P16050 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9957516 0.78 HSD17B10 (0.69) HSD17B10NPSR1CYP1A2CYP3A4HPGD
SCHEMBL9956376 0.71 HSD17B10 (0.42) HSD17B10NPSR1HPGDALDH1A1MAPT
SCHEMBL9956088 0.71 HSD17B10 (0.42) HSD17B10NPSR1CYP1A2CYP3A4HPGD
SCHEMBL13303521 0.68 ALDH1A1 (0.39) HSD17B10NPSR1CYP1A2CYP3A4HPGD
SCHEMBL11649419 0.61 HSD17B10 (1.00) HSD17B10NPSR1CYP1A2CYP3A4HPGD
SCHEMBL10818764 0.60 KMT2A (0.32) CYP3A4
SCHEMBL4163347 0.60 ALDH1A1 (0.39) ALDH1A1
SCHEMBL2154609 0.60 ALDH1A1 (0.39) ALDH1A1
SCHEMBL2162561 0.59 GABRA1 (0.50) HSD17B10CYP1A2CYP3A4HPGDKDM4E
Formaldehyde SCHEMBL26124284 0.59 HSD17B10 (0.61) HSD17B10NPSR1HPGDKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2655323-A1 INGENOL-3-ACYLATES III AND INGENOL-3-CARBAMATES LEO LABORATORIES LIMITED (IE) 2013-10-30 EP disclosed
WO-2012083953-A1 INGENOL-3-ACYLATES III AND INGENOL-3-CARBAMATES LEO PHARMA A/S (DK) 2012-06-28 WO disclosed