SCHEMBL9958887

SCHEMBL9958887

CC#CC(C)(C)C(=O)NC1C(=O)N(OCc2ccccc2)C(=O)c2ccccc21

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 6/20 0.38
PSEN2 P49810 6/20 0.38
APH1B Q8WW43 6/20 0.38
NCSTN Q92542 6/20 0.38
APH1A Q96BI3 6/20 0.38
PSENEN Q9NZ42 6/20 0.38
MAPT P10636 3/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
PPIA P62937 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
FFAR1 O14842 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
UBE2M P61081 1/20 0.32
DCUN1D1 Q96GG9 1/20 0.32
KCNA5 P22460 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9952711 0.87 ACHE (0.36) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL9953052 0.79 KCNA5 (0.36) MAPTMEN1KMT2AFFAR1TSHR
SCHEMBL9958850 0.74 MEN1 (0.43) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL9960452 0.73 KCNA5 (0.46) MAPTMEN1KMT2AKCNA5
SCHEMBL9958888 0.72 MEN1 (0.36) MAPTMEN1KMT2AALDH1A1FFAR1
SCHEMBL11787179 0.71 MEN1 (0.47) MAPTMEN1KMT2AALDH1A1FFAR1
SCHEMBL9959297 0.70 HDAC4 (0.49) MAPTMEN1KMT2AALDH1A1FFAR1
SCHEMBL9952002 0.69 MEN1 (0.45) MAPTMEN1KMT2AALDH1A1FFAR1
SCHEMBL10153741 0.69 ALDH1A1 (0.38) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL10153981 0.69 MEN1 (0.40) MAPTMEN1KMT2AALDH1A1FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085003-A1 2-HYDROXYISOQUINOLINE-1,3(2H,4H)-DIONES AND RELATED COMPOUNDS USEFUL AS HIV REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-06-28 WO claimed