SCHEMBL9960452

SCHEMBL9960452

CC(C)(C)NC(=O)C1C(=O)N(OCc2ccccc2)C(=O)c2ccccc21

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 13/20 0.46
KCNH2 Q12809 6/20 0.46
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9953052 0.89 KCNA5 (0.36) KCNA5KCNH2MEN1MAPTKMT2A
SCHEMBL9959297 0.86 HDAC4 (0.49) KCNA5MEN1MAPTKMT2A
SCHEMBL10153637 0.84 KCNA5 (0.42) KCNA5MEN1MAPTKMT2A
SCHEMBL9959313 0.84 KCNA5 (0.48) KCNA5MEN1MAPTKMT2A
SCHEMBL9958850 0.84 MEN1 (0.43) KCNA5MEN1MAPTKMT2A
SCHEMBL10153642 0.83 KCNA5 (0.42) KCNA5MEN1MAPTKMT2A
SCHEMBL11787179 0.83 MEN1 (0.47) MEN1MAPTKMT2A
SCHEMBL10153971 0.82 POLB (0.50) KCNA5MEN1MAPTKMT2A
SCHEMBL9958882 0.82 KMT2A (0.46) KCNA5KCNH2MEN1MAPTKMT2A
SCHEMBL9952002 0.81 MEN1 (0.45) MEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085003-A1 2-HYDROXYISOQUINOLINE-1,3(2H,4H)-DIONES AND RELATED COMPOUNDS USEFUL AS HIV REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-06-28 WO disclosed
WO-2012085003-A1 2-HYDROXYISOQUINOLINE-1,3(2H,4H)-DIONES AND RELATED COMPOUNDS USEFUL AS HIV REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-06-28 WO disclosed